SCHEMBL7273271

SCHEMBL7273271

O=C(O)C[C@@H]1C[C@@H](COC(c2ccccc2)(c2ccccc2)c2ccccc2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
TSHR P16473 1/20 0.40
CHRM3 P20309 3/20 0.35
MEN1 O00255 2/20 0.34
CYP1A2 P05177 2/20 0.34
CYP3A4 P08684 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
KMT2A Q03164 2/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
ALOX12 P18054 1/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ITGB3 P05106 1/20 0.33
ITGA2B P08514 1/20 0.33
ITGB1 P05556 1/20 0.33
ITGA5 P08648 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275757 0.89 SMN1; SMN2 (0.39) ALDH1A1SMN1; SMN2TSHRCHRM3LMNA
SCHEMBL7272646 0.88 GSK3A (0.35) ALDH1A1CHRM3MEN1KMT2AGSK3A
SCHEMBL7275231 0.84 CHRNB4 (0.37) ALDH1A1CHRM3MEN1KMT2AGSK3A
SCHEMBL7283097 0.84 HRH3 (0.40) TSHRMEN1CYP3A4CYP2D6CYP2C9
SCHEMBL7275948 0.84 CHRNB4 (0.37) ALDH1A1CHRM3MEN1KMT2AGSK3A
SCHEMBL7276102 0.83 FAAH (0.38) GSK3AGSK3B
SCHEMBL7275115 0.83 SIGMAR1 (0.39) ALDH1A1MEN1KMT2AGSK3AGSK3B
SCHEMBL7282778 0.82 FAAH (0.39) GSK3AGSK3B
SCHEMBL7276617 0.82 FAAH (0.37) TSHRCHRM3MEN1CYP1A2CYP3A4
SCHEMBL7282531 0.81 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2TSHRMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed