SCHEMBL7273697

SCHEMBL7273697

C=CC[C@@H]1C[C@@H](COC(c2ccccc2)(c2ccccc2)c2ccccc2)N(CCc2ccc3ccccc3c2)C1=O

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.34
SLC6A4 P31645 1/20 0.33
CHRM3 P20309 1/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
ELANE P08246 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
ALDH1A1 P00352 1/20 0.30
THRB P10828 1/20 0.30
TP53 P04637 1/20 0.30
MDM2 Q00987 1/20 0.30
CYP1A2 P05177 1/20 0.30
ACHE P22303 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7282618 0.89 ALDH1A1 (0.34) HCRTR1HCRTR2SIGMAR1ALDH1A1TP53
SCHEMBL7275231 0.84 CHRNB4 (0.37) CHRM3ELANESIGMAR1ALDH1A1TP53
SCHEMBL7275948 0.84 CHRNB4 (0.37) CHRM3ELANESIGMAR1ALDH1A1TP53
SCHEMBL7279479 0.83 MAPT (0.36)
SCHEMBL7274612 0.83 HRH3 (0.36) HRH3SLC6A4HCRTR1HCRTR2ELANE
SCHEMBL7276617 0.83 FAAH (0.37) CHRM3ELANESIGMAR1TP53CYP1A2
SCHEMBL7284852 0.82 HRH3 (0.40) HRH3SLC6A4HCRTR1HCRTR2SIGMAR1
SCHEMBL7283004 0.82 SLC6A4 (0.40) HRH3SLC6A4CYP1A2
SCHEMBL7281843 0.81 EHMT2 (0.35) ALDH1A1TP53MDM2
SCHEMBL7283379 0.80 SSTR5 (0.41) HRH3SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed