SCHEMBL7274612

SCHEMBL7274612

C=CC[C@@H]1C[C@@H](COS(C)(=O)=O)N(CCc2ccc3ccccc3c2)C1=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.36
HCRTR1 O43613 2/20 0.35
HCRTR2 O43614 2/20 0.35
SLC6A4 P31645 3/20 0.34
ELANE P08246 2/20 0.33
BACE1 P56817 1/20 0.33
HDAC3 O15379 2/20 0.32
HDAC4 P56524 2/20 0.32
HDAC1 Q13547 2/20 0.32
HDAC7 Q8WUI4 2/20 0.32
HDAC2 Q92769 2/20 0.32
HDAC10 Q969S8 2/20 0.32
HDAC11 Q96DB2 2/20 0.32
HDAC8 Q9BY41 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
HDAC5 Q9UQL6 2/20 0.32
HDAC9 Q9UKV0 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A3 Q01959 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281928 0.88 F2 (0.36) HCRTR1HCRTR2ELANEKCNH2SIGMAR1
SCHEMBL7284852 0.84 HRH3 (0.40) HRH3HCRTR1HCRTR2SLC6A4BACE1
SCHEMBL7283004 0.84 SLC6A4 (0.40) HRH3SLC6A4HDAC3HDAC4HDAC1
SCHEMBL7273697 0.83 HRH3 (0.34) HRH3HCRTR1HCRTR2SLC6A4ELANE
SCHEMBL7274544 0.83 MAPT (0.39) ALDH1A1
SCHEMBL7274866 0.82 CHRNB4 (0.38) ELANEKCNH2SIGMAR1F2CTSG
SCHEMBL7275714 0.81 FAAH (0.39) ELANEF2CTSG
SCHEMBL7272678 0.80 HRH3 (0.36) HRH3HCRTR1HCRTR2SLC6A4HDAC3
SCHEMBL7273490 0.79 F2 (0.37) HCRTR2ELANEALDH1A1F2CTSG
SCHEMBL7281067 0.79 MGLL (0.41) HRH3KCNH2SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed