SCHEMBL7274028

SCHEMBL7274028

CCc1cn(C(=O)NC2CC3CCC(C2)N3C)c2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 9/20 0.56
TMEM97 Q5BJF2 1/20 0.56
SIGMAR1 Q99720 1/20 0.56
HTR4 Q13639 1/20 0.56
ALDH1A1 P00352 1/20 0.53
CYP3A4 P08684 1/20 0.53
TSHR P16473 1/20 0.53
MAPK1 P28482 1/20 0.53
HSD17B10 Q99714 1/20 0.53
HTR3E A5X5Y0 5/20 0.52
HTR3B O95264 5/20 0.52
HTR3D Q70Z44 5/20 0.52
HTR3C Q8WXA8 5/20 0.52
SLC22A2 O15244 1/20 0.48
CHRNB2 P17787 1/20 0.48
CHRNA3 P32297 1/20 0.48
CHRNA4 P43681 1/20 0.48
KCNH2 Q12809 1/20 0.48
SLC47A1 Q96FL8 1/20 0.48
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7435410 0.99 HTR3A (0.55) HTR3ATMEM97SIGMAR1HTR4ALDH1A1
SCHEMBL7267718 0.86 ALDH1A1 (0.55) HTR3ATMEM97SIGMAR1HTR4ALDH1A1
Hydrochloric Acid SCHEMBL7443261 0.85 ALDH1A1 (0.54) HTR3ATMEM97SIGMAR1HTR4ALDH1A1
SCHEMBL9602256 0.82 ALDH1A1 (0.51) HTR3ATMEM97SIGMAR1HTR4ALDH1A1
SCHEMBL7266776 0.76 HTR3A (0.55) HTR3ATMEM97SIGMAR1HTR4ALDH1A1
Hydrochloric Acid SCHEMBL7429564 0.75 HTR3A (0.54) HTR3ATMEM97SIGMAR1HTR4ALDH1A1
SCHEMBL9478363 0.73 DRD2 (0.42) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL1041383 0.72 HTR4 (1.00) HTR3ATMEM97SIGMAR1HTR4HTR3E
SCHEMBL6669870 0.72 HTR4 (1.00) HTR3ATMEM97SIGMAR1HTR4HTR3E
SCHEMBL7343018 0.71 HTR3A (0.85) HTR3ATMEM97SIGMAR1HTR4HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0278173-B1 Use of heterocyclic derivatives in the treatment of depressions GLAXO GROUP LTD (GB) 1993-11-03 EP claimed
EP-0247266-B1 INDOLE DERIVATIVES HAVING AN AZABICYCLIC SIDE CHAIN, PROCESS FOR THEIR PREPARATION, INTERMEDIATES, AND PHARMACEUTICAL COMPOSITIONS BEECHAM GROUP PLC (GB) 1993-03-10 EP claimed
EP-0247266-A1 Indole derivatives having an azabicyclic side chain, process for their preparation, intermediates, and pharmaceutical compositions BEECHAM GROUP PLC (GB) 1987-12-02 EP claimed
EP-0278173-B1 Use of heterocyclic derivatives in the treatment of depressions GLAXO GROUP LTD (GB) 1993-11-03 EP disclosed