SCHEMBL7274068

SCHEMBL7274068

N=C(N)NCCc1ccc(C(=O)NC[C@@H]2C[C@@H](CC(=O)O)C(=O)N2CCCc2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.42
F2 P00734 5/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
RAB9A P51151 5/20 0.38
NPC1 O15118 4/20 0.38
ITGB3 P05106 3/20 0.37
ITGA2B P08514 3/20 0.37
CHRM4 P08173 1/20 0.37
LMNA P02545 1/20 0.37
HPGD P15428 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
F10 P00742 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
GAA P10253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7276505 0.93 F2 (0.41) KDM1AF2HDAC2HDAC8HDAC6
SCHEMBL7272267 0.93 F10 (0.41) KDM1AHDAC2HDAC8HDAC6RAB9A
SCHEMBL7282394 0.88 ITGB3 (0.44) KDM1AHDAC8HDAC6RAB9ANPC1
SCHEMBL7284039 0.88 ITGB3 (0.42) KDM1AHDAC8HDAC6RAB9ANPC1
Water SCHEMBL7273367 0.88 F10 (0.45) F2ITGB3ITGA2BF10
SCHEMBL7282719 0.87 KDM1A (0.38) KDM1AITGB3ITGA2BCHRM4LMNA
SCHEMBL7274533 0.86 TSHR (0.40) F2ITGB3ITGA2BLMNAMEN1
Water SCHEMBL7281948 0.86 PPARG (0.41) KDM1AF2ITGB3ITGA2BF10
SCHEMBL7274469 0.85 LMNA (0.42) F2HDAC2HDAC8HDAC6ITGB3
SCHEMBL7274776 0.85 ITGB3 (0.45) ITGB3ITGA2BF10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed