SCHEMBL7274141

SCHEMBL7274141

C=CC[C@@H]1C[C@@H](COc2ccc(C(=O)Nc3ccc(C#N)cc3)cc2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
LMNA P02545 3/20 0.40
MAPT P10636 3/20 0.40
NAMPT P43490 2/20 0.40
NR1H4 Q96RI1 1/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
CYP19A1 P11511 1/20 0.38
PGR P06401 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
HDAC1 Q13547 1/20 0.37
CYSLTR1 Q9Y271 2/20 0.37
POLB P06746 1/20 0.36
ABCB1 P08183 1/20 0.36
HPGD P15428 1/20 0.36
ABCG2 Q9UNQ0 1/20 0.36
KCNA5 P22460 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7276118 1.00 ALDH1A1 (0.40) ALDH1A1LMNAMAPTNAMPTNR1H4
SCHEMBL7284072 0.90 ALDH1A1 (0.43) ALDH1A1LMNAMAPTNAMPTNR1H4
SCHEMBL7284876 0.88 ALDH1A1 (0.43) ALDH1A1LMNAMAPTNAMPTNR1H4
SCHEMBL7274156 0.87 ABCB1 (0.42) MEN1KMT2AABCB1HPGDABCG2
SCHEMBL7282764 0.87 ABCB1 (0.42) MEN1KMT2AABCB1HPGDABCG2
SCHEMBL7283159 0.87 ABCB1 (0.42) MEN1KMT2AABCB1HPGDABCG2
SCHEMBL7275535 0.85 CCR3 (0.43) ALDH1A1LMNANAMPTHDAC1
SCHEMBL7273502 0.85 AR (0.51) MAPTCYP19A1PGRMEN1KMT2A
SCHEMBL7282205 0.84 ABCB1 (0.41) MEN1KMT2AABCB1HPGDABCG2
SCHEMBL7281199 0.83 SLC6A2 (0.37) ALDH1A1LMNAMAPTNAMPTABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed