SCHEMBL7284072

SCHEMBL7284072

N#Cc1ccc(NC(=O)c2ccc(OC[C@@H]3C[C@@H](CC(=O)O)C(=O)N3CCCc3ccccc3)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
LMNA P02545 3/20 0.43
MAPT P10636 1/20 0.43
NAMPT P43490 2/20 0.41
NR1H4 Q96RI1 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.41
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
CYP19A1 P11511 1/20 0.40
PGR P06401 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
HDAC1 Q13547 1/20 0.39
CYSLTR1 Q9Y271 2/20 0.38
PTGIR P43119 1/20 0.38
KCNA5 P22460 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7284876 0.93 ALDH1A1 (0.43) ALDH1A1LMNAMAPTNAMPTNR1H4
SCHEMBL7276118 0.90 ALDH1A1 (0.40) ALDH1A1LMNAMAPTNAMPTNR1H4
SCHEMBL7274141 0.90 ALDH1A1 (0.40) ALDH1A1LMNAMAPTNAMPTNR1H4
SCHEMBL7275113 0.90 ITGB3 (0.48) ALDH1A1LMNAMAPTNR1H4NPC1
SCHEMBL7276310 0.90 ITGB3 (0.48) ALDH1A1LMNAMAPTNR1H4NPC1
SCHEMBL7276469 0.88 ABCB1 (0.45) ALDH1A1LMNAMAPTSMN1; SMN2MEN1
SCHEMBL7275504 0.88 ABCB1 (0.45) ALDH1A1LMNAMAPTSMN1; SMN2MEN1
SCHEMBL7273402 0.86 ABCB1 (0.44) ALDH1A1LMNAMAPTNAMPTMEN1
SCHEMBL7283466 0.84 PPARA (0.40) ALDH1A1LMNAMAPTNAMPTSMN1; SMN2
SCHEMBL7274964 0.84 CCR3 (0.44) ALDH1A1NAMPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed