SCHEMBL7274240

SCHEMBL7274240

CC1(C)Oc2ccc(C#N)cc2C(Oc2ccccn2)C1O

nearest known ligand 0.62

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 8/20 0.62
ABCB1 P08183 7/20 0.50
KDM4E B2RXH2 1/20 0.47
CYP3A4 P08684 1/20 0.46
ALOX15 P16050 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7360393 0.86 ABCC9 (0.58) ABCC9ABCB1KDM4ECYP3A4
SCHEMBL7331034 0.86 ABCC9 (0.56) ABCC9ABCB1KDM4ECYP3A4
SCHEMBL7330523 0.86 ABCC9 (0.56) ABCC9ABCB1KDM4ECYP3A4
SCHEMBL7357182 0.84 ABCC9 (0.45) ABCC9ABCB1KDM4ECYP3A4ALOX15
SCHEMBL8088840 0.84 ABCC9 (0.56) ABCC9ABCB1KDM4ECYP3A4
SCHEMBL7360016 0.83 ABCC9 (0.44) ABCC9ABCB1KDM4ECYP3A4ALOX15
SCHEMBL8085199 0.83 ABCC9 (0.42) ABCC9ABCB1
SCHEMBL8084989 0.83 ABCC9 (0.57) ABCC9ABCB1KDM4ECYP3A4ALOX15
SCHEMBL7331710 0.82 ABCC9 (0.58) ABCC9ABCB1KDM4ECYP3A4
SCHEMBL7325382 0.82 ABCC9 (0.54) ABCC9ABCB1KDM4ECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0363883-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1990-04-18 EP disclosed
EP-0346724-A1 Chroman derivates MERCK PATENT GmbH (DE) 1989-12-20 EP disclosed