SCHEMBL7360016

SCHEMBL7360016

N#Cc1ccc2c(c1)C(Oc1ccccn1)C(O)C1(CCCCC1)O2

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 9/20 0.44
ABCB1 P08183 4/20 0.36
AVPR1A P37288 1/20 0.35
ABCC8 Q09428 2/20 0.35
KCNJ11 Q14654 2/20 0.35
KCNJ8 Q15842 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 1/20 0.35
CYP3A4 P08684 1/20 0.34
ALOX15 P16050 1/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7357182 0.99 ABCC9 (0.45) ABCC9ABCB1AVPR1AABCC8KCNJ11
SCHEMBL7274240 0.83 ABCC9 (0.62) ABCC9ABCB1CYP3A4ALOX15KDM4E
SCHEMBL7355509 0.82 ABCC9 (0.40) ABCC9ABCB1ABCC8KCNJ11KCNJ8
SCHEMBL8088457 0.81 ABCC9 (0.40) ABCC9ABCB1ABCC8KCNJ11KCNJ8
SCHEMBL7364124 0.81 ABCC9 (0.41) ABCC9ABCB1ABCC8KCNJ11KCNJ8
SCHEMBL8084932 0.80 ABCC9 (0.40) ABCC9ABCB1ABCC8KCNJ11KCNJ8
SCHEMBL9876186 0.76 ABCC9 (0.41) ABCC9ABCB1ABCC8KCNJ11KCNJ8
SCHEMBL9876177 0.76 ABCC9 (0.41) ABCC9ABCB1ABCC8KCNJ11KCNJ8
SCHEMBL9876183 0.76 ABCC9 (0.41) ABCC9ABCB1ABCC8KCNJ11KCNJ8
SCHEMBL9529091 0.73 ABCC9 (0.42) ABCC9ABCB1ABCC8KCNJ11KCNJ8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0363883-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1990-04-18 EP disclosed