SCHEMBL8085199

SCHEMBL8085199

CC1(C)Oc2ccc(Br)cc2C(Oc2ccccn2)C1O

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 6/20 0.42
KCNE1 P15382 3/20 0.33
KCNQ1 P51787 3/20 0.33
AVPR1A P37288 1/20 0.33
HTR2B P41595 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
ABCB1 P08183 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7274240 0.83 ABCC9 (0.62) ABCC9ABCB1
SCHEMBL8085013 0.82 ABCC9 (0.41) ABCC9NPC1RAB9A
SCHEMBL8088486 0.81 ABCC9 (0.42) ABCC9NPC1RAB9A
SCHEMBL9589063 0.81 ABCC9 (0.48) ABCC9KCNE1KCNQ1ABCB1
SCHEMBL9589058 0.81 ABCC9 (0.48) ABCC9KCNE1KCNQ1ABCB1
SCHEMBL9589053 0.81 ABCC9 (0.48) ABCC9KCNE1KCNQ1ABCB1
SCHEMBL7324168 0.79 ABCC9 (0.38) ABCC9KCNE1KCNQ1
SCHEMBL7330531 0.79 ABCC9 (0.38) ABCC9KCNE1KCNQ1
SCHEMBL8076897 0.78 ABCC9 (0.38) ABCC9KCNE1KCNQ1
SCHEMBL9565062 0.76 TP53 (0.34) AVPR1ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed