SCHEMBL7274397

SCHEMBL7274397

CCOC(=O)[C@H](Cc1cc(I)c(Sc2ccc(OC)c(Cc3ccc(OC)cc3)c2)c(I)c1)NC(=O)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
PDE2A O00408 5/20 0.36
EPHX2 P34913 1/20 0.34
PPARG P37231 1/20 0.34
CAPN1 P07384 1/20 0.33
MAPT P10636 1/20 0.33
PPARD Q03181 1/20 0.33
PPARA Q07869 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7285771 0.89 ALDH1A1 (0.33) ALDH1A1PDE2APPARDPPARA
SCHEMBL7274092 0.89 ALDH1A1 (0.53) ALDH1A1PDE2AMAPT
SCHEMBL7273900 0.81 ALDH1A1 (0.33) ALDH1A1PDE2APPARDPPARA
SCHEMBL7285392 0.79 ALDH1A1 (0.44) ALDH1A1
SCHEMBL5114514 0.70 MME (0.45) ALDH1A1
SCHEMBL5110447 0.70 MME (0.45) ALDH1A1
SCHEMBL8731461 0.69 THRB (0.51) ALDH1A1PPARGMAPT
SCHEMBL5114432 0.67 MDM4 (0.42) ALDH1A1MAPT
SCHEMBL5549364 0.67 MDM4 (0.42) ALDH1A1MAPT
SCHEMBL8730077 0.67 BACE1 (0.43) EPHX2PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5061798-A Intermediates in the formation of synthetic hormones, mimic effects of thyroid hormones; little or no effect on the heart SMITH KLINE & FRENCH LABORATORIES, LTD. (GB) 1991-10-29 US disclosed
EP-0188351-B1 CHEMICAL COMPOUNDS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-03-13 EP disclosed
US-4910305-A Containing a protected 4-hydroxyphenyl SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1990-03-20 US disclosed
US-4826876-A WITHOUT EFFECT ON HEART SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1989-05-02 US disclosed
US-4766121-A NOT AFFECTING THE HEART SMITH KLINE & FRENCH LABORATORIES LTD. (GB) 1988-08-23 US disclosed
EP-0188351-A2 Chemical compounds SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1986-07-23 EP disclosed