SCHEMBL7285771

SCHEMBL7285771

CCOC(=O)[C@H](Cc1cc(I)c(Sc2ccc(OC)c(Cc3ccc(OC)nc3)c2)c(I)c1)NC(=O)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.33
PDE2A O00408 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31
NR3C1 P04150 1/20 0.31
OPRK1 P41145 1/20 0.30
KLKB1 P03952 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
PDE5A O76074 2/20 0.30
PDE6D O43924 1/20 0.30
PDE6A P16499 1/20 0.30
PDE6G P18545 1/20 0.30
PDE6B P35913 1/20 0.30
PDE6C P51160 1/20 0.30
PDE6H Q13956 1/20 0.30
ACACB O00763 1/20 0.30
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273900 0.92 ALDH1A1 (0.33) ALDH1A1PDE2APPARDPPARANR3C1
SCHEMBL7285392 0.90 ALDH1A1 (0.44) ALDH1A1MEN1KMT2A
SCHEMBL7274397 0.89 ALDH1A1 (0.41) ALDH1A1PDE2APPARDPPARA
SCHEMBL7273661 0.85 FOLH1 (0.37) KLKB1
SCHEMBL7274092 0.79 ALDH1A1 (0.53) ALDH1A1PDE2AMEN1KMT2A
SCHEMBL7281994 0.69 ALDH1A1 (0.41) ALDH1A1PDE5APDE6DPDE6APDE6G
SCHEMBL10413380 0.69 CYP1A2 (0.33) ALDH1A1MEN1KMT2A
SCHEMBL7282033 0.68 TUBB4A (0.40)
SCHEMBL10563236 0.68 ALDH1A1 (0.39) ALDH1A1PDE5APDE6DPDE6APDE6G
SCHEMBL5114432 0.65 MDM4 (0.42) ALDH1A1NR3C1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5061798-A Intermediates in the formation of synthetic hormones, mimic effects of thyroid hormones; little or no effect on the heart SMITH KLINE & FRENCH LABORATORIES, LTD. (GB) 1991-10-29 US disclosed
EP-0188351-B1 CHEMICAL COMPOUNDS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-03-13 EP disclosed
US-4910305-A Containing a protected 4-hydroxyphenyl SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1990-03-20 US disclosed
US-4826876-A WITHOUT EFFECT ON HEART SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1989-05-02 US disclosed
US-4766121-A NOT AFFECTING THE HEART SMITH KLINE & FRENCH LABORATORIES LTD. (GB) 1988-08-23 US disclosed
EP-0188351-A2 Chemical compounds SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1986-07-23 EP disclosed