SCHEMBL7274964

SCHEMBL7274964

N#Cc1ccc(C(=O)NC[C@@H]2C[C@@H](CC(=O)O)C(=O)N2CCCc2ccccc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 1/20 0.44
MAOA P21397 2/20 0.42
NAMPT P43490 3/20 0.42
SIGMAR1 Q99720 2/20 0.41
CHRM4 P08173 2/20 0.41
TMEM97 Q5BJF2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TSHR P16473 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
OPRM1 P35372 2/20 0.39
HTR1A P08908 1/20 0.39
DRD4 P21917 1/20 0.39
HTR2A P28223 1/20 0.39
HRH1 P35367 1/20 0.39
CTSL P07711 2/20 0.39
CTSB P07858 2/20 0.39
CTSK P43235 2/20 0.39
KDM1A O60341 2/20 0.39
HDAC6 Q9UBN7 2/20 0.39
EPHX2 P34913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7281678 0.90 HTR1A (0.42) MAOANAMPTALDH1A1TSHRSMN1; SMN2
SCHEMBL7274708 0.89 CHRM4 (0.42) CCR3MAOANAMPTSIGMAR1CHRM4
Methyl Alcohol SCHEMBL8879759 0.89 HTR1A (0.40) CCR3NAMPTCHRM4HTR1AKDM1A
SCHEMBL7275535 0.89 CCR3 (0.43) CCR3MAOANAMPTSIGMAR1CHRM4
SCHEMBL7274088 0.88 HTR1A (0.42) NAMPTALDH1A1TSHRSMN1; SMN2OPRM1
SCHEMBL7282394 0.87 ITGB3 (0.44) CHRM4ALDH1A1TSHRSMN1; SMN2OPRM1
SCHEMBL7284039 0.87 ITGB3 (0.42) CHRM4ALDH1A1TSHRSMN1; SMN2OPRM1
Water SCHEMBL7273367 0.85 F10 (0.45)
SCHEMBL7277147 0.84 ASAH1 (0.42) CHRM4ALDH1A1TSHRSMN1; SMN2OPRM1
SCHEMBL7280929 0.84 KDM1A (0.42) MAOANAMPTCHRM4ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed