SCHEMBL7275250

SCHEMBL7275250

COc1ccc(-n2ccc[c]c2=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.53
MAPT P10636 3/20 0.44
LMNA P02545 2/20 0.44
KDM4E B2RXH2 2/20 0.44
HTT P42858 2/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MGLL Q99685 1/20 0.44
POLB P06746 1/20 0.43
PKM P14618 2/20 0.41
F10 P00742 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HCAR1 Q9BXC0 1/20 0.40
G6PD P11413 1/20 0.40
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
ELANE P08246 1/20 0.39
NR1H3 Q13133 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10946472 0.77 ATM (0.44) ALDH1A1MAPTLMNAKDM4EHTT
SCHEMBL2115832 0.77 F10 (0.59) ALDH1A1MAPTLMNAKDM4EHTT
SCHEMBL25541378 0.71 ALDH1A1 (0.59) ALDH1A1MAPTLMNAKDM4EHTT
SCHEMBL8461478 0.69 CA12 (0.42) ALDH1A1MAPTLMNAHTTSMN1; SMN2
SCHEMBL6282109 0.68 ALDH1A1 (0.56) ALDH1A1MAPTLMNAKDM4EHTT
SCHEMBL14280098 0.68 ALDH1A1 (0.47) ALDH1A1MAPTLMNAKDM4EHTT
SCHEMBL1727656 0.68 LTA4H (0.60) ALDH1A1MAPTLMNAHTTMGLL
SCHEMBL1494699 0.68 ALDH1A1 (0.55) ALDH1A1MAPTLMNAKDM4EHTT
SCHEMBL15328181 0.67 ALDH1A1 (0.50) ALDH1A1MAPTLMNAKDM4EHTT
SCHEMBL8718494 0.67 HCAR1 (0.51) ALDH1A1MAPTLMNAHTTMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0418696-A2 Derivatives of aminoacids MERCK PATENT GmbH (DE) 1991-03-27 EP disclosed
EP-0401507-A1 Cyclic agonists of tachykinin MERCK PATENT GmbH (DE) 1990-12-12 EP disclosed
EP-0284942-A2 Amino-acid derivatives MERCK PATENT GmbH (DE) 1988-10-05 EP disclosed
EP-0272444-A2 Renin-inhibiting peptides MERCK PATENT GmbH (DE) 1988-06-29 EP disclosed
EP-0264795-A2 Amino acid derivatives MERCK PATENT GmbH (DE) 1988-04-27 EP disclosed