SCHEMBL7275576

SCHEMBL7275576

N#Cc1ccc(-c2ccc(O)c(C(F)(F)F)c2)cc1

nearest known ligand 0.63

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 3/20 0.63
AR P10275 6/20 0.57
P4HB P07237 2/20 0.53
HSD17B1 P14061 2/20 0.50
HSD17B2 P37059 2/20 0.50
MMP3 P08254 1/20 0.50
CYP19A1 P11511 1/20 0.48
PGR P06401 2/20 0.48
PTPN5 P54829 1/20 0.45
PDK2 Q15119 1/20 0.44
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
RXRG P48443 1/20 0.44
TRPV4 Q9HBA0 1/20 0.44
GYS1 P13807 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL524173 0.87 P4HB (0.56) KIF11ARP4HBHSD17B1HSD17B2
SCHEMBL1938893 0.83 HSD17B1 (0.65) KIF11ARHSD17B1HSD17B2PGR
SCHEMBL29485676 0.83 HSD17B1 (0.65) KIF11ARHSD17B1HSD17B2PGR
SCHEMBL397926 0.81 KIF11 (0.65) KIF11ARMMP3PGRPTPN5
SCHEMBL4049024 0.79 KIF11 (0.63) KIF11ARMMP3PGRPTPN5
SCHEMBL27546220 0.78 HSD17B1 (0.60) KIF11ARHSD17B1HSD17B2MMP3
SCHEMBL9063141 0.77 KIF11 (0.59) KIF11ARP4HBHSD17B1HSD17B2
SCHEMBL2786052 0.77 KIF11 (0.59) KIF11ARP4HBHSD17B1HSD17B2
SCHEMBL7283993 0.76 KIF11 (0.58) KIF11ARPGR
SCHEMBL28668535 0.75 KIF11 (0.57) KIF11ARP4HBPGRPTPN5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
US-5541343-A ANTIAGGLOMERANTS FOR CELLS OR ANTICOAGULANTS KARL THOMAE GMBH (DE) 1996-07-30 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed