SCHEMBL7276136

SCHEMBL7276136

C=CC[C@@H]1C[C@@H](CNC(=O)c2ccc3c(c2)CC(CNC(=O)OC(C)(C)C)C3)N(CCCc2ccccc2)C1=O

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.40
ACACB O00763 6/20 0.40
ACACA Q13085 5/20 0.40
DRD2 P14416 2/20 0.35
KDM4E B2RXH2 1/20 0.35
PKM P14618 1/20 0.35
DRD3 P35462 1/20 0.35
HTR1A P08908 2/20 0.34
OPRM1 P35372 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
BRD4 O60885 1/20 0.34
NAMPT P43490 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7272709 0.92 SIGMAR1 (0.38) SIGMAR1ACACBACACADRD2DRD3
SCHEMBL7284329 0.91 ACACB (0.41) SIGMAR1ACACBACACAKDM4EPKM
SCHEMBL8881851 0.90 SIGMAR1 (0.38) SIGMAR1ACACBACACADRD2DRD3
SCHEMBL7273654 0.88 SIGMAR1 (0.44) SIGMAR1DRD2DRD3OPRM1NAMPT
SCHEMBL7280539 0.87 SIGMAR1 (0.44) SIGMAR1ACACBACACADRD2DRD3
SCHEMBL7283282 0.85 KDM4E (0.41) SIGMAR1DRD2KDM4EPKMHTR1A
SCHEMBL7274101 0.84 ITGB3 (0.41) SIGMAR1ACACBACACAOPRM1NAMPT
SCHEMBL7304783 0.83 SIGMAR1 (0.39) SIGMAR1DRD2KDM4EPKMDRD3
SCHEMBL7271758 0.82 SIGMAR1 (0.38) SIGMAR1ACACBACACAHTR1AOPRM1
SCHEMBL7272740 0.81 SIGMAR1 (0.37) SIGMAR1DRD2DRD3NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed