SCHEMBL7280539

SCHEMBL7280539

C=CC[C@@H]1C[C@@H](CNC(=O)c2cccc(CCNC(=O)OC(C)(C)C)c2)N(CCCc2ccccc2)C1=O

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.44
DRD2 P14416 2/20 0.43
DRD3 P35462 1/20 0.40
HTR1A P08908 2/20 0.39
NAMPT P43490 3/20 0.38
ACACB O00763 1/20 0.38
ACACA Q13085 1/20 0.38
MAOA P21397 1/20 0.37
SLC5A7 Q9GZV3 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
FAAH O00519 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7273654 0.93 SIGMAR1 (0.44) SIGMAR1DRD2DRD3NAMPTNPC1
SCHEMBL7272424 0.91 SIGMAR1 (0.45) SIGMAR1DRD2HTR1ANAMPTACACB
SCHEMBL7276136 0.87 SIGMAR1 (0.40) SIGMAR1DRD2DRD3HTR1ANAMPT
SCHEMBL7283982 0.86 SIGMAR1 (0.43) SIGMAR1NAMPTACACBFAAH
SCHEMBL7272709 0.85 SIGMAR1 (0.38) SIGMAR1DRD2DRD3HTR1ANAMPT
SCHEMBL7304783 0.84 SIGMAR1 (0.39) SIGMAR1DRD2DRD3FAAH
SCHEMBL7274528 0.84 SIGMAR1 (0.45) SIGMAR1NAMPTNPC1RAB9A
SCHEMBL7280624 0.83 SIGMAR1 (0.45) SIGMAR1NAMPTFAAH
SCHEMBL7274557 0.83 SIGMAR1 (0.44) SIGMAR1ACACB
SCHEMBL7275472 0.82 SIGMAR1 (0.41) SIGMAR1DRD2DRD3NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5621103-A 3-(SUBSTITUTED METHYLAMINOCARBONYL)-1,2,3,4-TETRAHYDRO-(1)BENZOTHIENO(2,3-C) PYRIDINES; ANXIOLYTIC AGENTS; LEARNING ENHANCEMENT ASAHI KASEI KOGYO KABUSHIKI KAISHA (JP) 1997-04-15 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed