SCHEMBL7276441

SCHEMBL7276441

COc1ccc(-c2ccc(NC(=O)OCc3ccccc3)c(=O)[nH]2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
KDM4E B2RXH2 1/20 0.51
GAA P10253 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
RXFP1 Q9HBX9 1/20 0.51
TACR3 P29371 1/20 0.50
NPC1 O15118 3/20 0.49
RAB9A P51151 2/20 0.49
ELANE P08246 2/20 0.47
ATM Q13315 2/20 0.46
MMP1 P03956 1/20 0.45
MMP9 P14780 1/20 0.45
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ACHE P22303 1/20 0.44
PTPN1 P18031 1/20 0.44
CASP3 P42574 1/20 0.44
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6556065 0.90 NPC1 (0.53) ALDH1A1KDM4ESMN1; SMN2TACR3NPC1
SCHEMBL7276750 0.88 RAB9A (0.48) ALDH1A1GAANPC1RAB9AELANE
SCHEMBL7276640 0.81 MGLL (0.46) ALDH1A1KDM4ESMN1; SMN2TACR3NPC1
SCHEMBL4416727 0.78 NPC1 (0.62) ALDH1A1SMN1; SMN2NPC1RAB9AMMP1
SCHEMBL1330921 0.77 CASP3 (0.51) SMN1; SMN2NPC1RAB9AELANEPTPN1
SCHEMBL7342183 0.76 NPC1 (0.56) ALDH1A1SMN1; SMN2NPC1RAB9AMMP1
SCHEMBL5113764 0.75 NPC1 (0.54) ALDH1A1SMN1; SMN2NPC1RAB9AELANE
SCHEMBL1223807 0.75 RAB9A (0.67) ALDH1A1GAASMN1; SMN2NPC1RAB9A
SCHEMBL8401148 0.75 TACR3 (0.46) ALDH1A1KDM4ESMN1; SMN2TACR3NPC1
SCHEMBL11261916 0.75 KDM4E (0.57) ALDH1A1KDM4EGAASMN1; SMN2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0509769-B1 Heterocyclic amides having HLE inhibiting activity ZENECA LTD (GB) 1996-09-11 EP disclosed
US-5521179-A Heterocyclic amides ZENECA LIMITED (GB) 1996-05-28 US disclosed
EP-0509769-A2 Heterocyclic amides having HLE inhibiting activity ZENECA LIMITED (GB) 1992-10-21 EP disclosed