SCHEMBL7277572

SCHEMBL7277572

CN(C)CCC(Cc1ccccc1)C(=O)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.50
UBE2N P61088 1/20 0.49
CHRM1 P11229 1/20 0.48
FOLH1 Q04609 2/20 0.47
HPGD P15428 1/20 0.46
CPA3 P15088 3/20 0.46
CPA1 P15085 2/20 0.45
CPB1 P15086 1/20 0.45
CPB2 Q96IY4 1/20 0.45
HTR2A P28223 1/20 0.44
HRH1 P35367 1/20 0.44
UTS2R Q9UKP6 2/20 0.43
TAAR1 Q96RJ0 1/20 0.43
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6249330 0.84 CCR1 (0.50) CYP1A2UBE2NCHRM1FOLH1HPGD
SCHEMBL620307 0.78 CYP1A2 (0.64) CYP1A2FOLH1CPA3CPA1CPB1
SCHEMBL10010707 0.77 FOLH1 (0.69) CYP1A2UBE2NCHRM1FOLH1CPA3
SCHEMBL7277645 0.75 MTNR1A (0.55) CYP1A2CPA3
Acetamide SCHEMBL7277641 0.72 CYP1A2 (0.56) CYP1A2FOLH1CPA3CPA1CPB1
SCHEMBL25218779 0.72 ACHE (0.56) HPGD
SCHEMBL26730248 0.72 HTR2A (0.53) UBE2NCHRM1HTR2AHRH1TAAR1
SCHEMBL8572290 0.71 CYP1A2 (0.55) CYP1A2UBE2NFOLH1HPGDCPA3
SCHEMBL38656098 0.71 CYP1A2 (0.59) CYP1A2FOLH1CPA3CPA1CPB1
SCHEMBL6698882 0.71 CYP1A2 (0.54) CYP1A2UBE2NCHRM1FOLH1CPA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4766110-A INHIBITS ANGIOTENSIN CONVERTING ENZYME, HYPOTENSIVE AGENTS RYAN JAMES W (US) 1988-08-23 US disclosed
EP-0073143-B1 NOVEL COMPLEX AMIDO AND IMIDO DERIVATIVES OF CARBOXYALKYL PEPTIDES AND THIOETHERS AND ETHERS OF PEPTIDES Ryan, James Walter (US) 1985-11-21 EP disclosed
EP-0073143-A2 Novel complex amido and imido derivatives of carboxyalkyl peptides and thioethers and ethers of peptides Ryan, James Walter (US) 1983-03-02 EP disclosed
EP-0048159-A2 Novel carboxyalkyl peptides and thioethers and ethers of peptides as antihypertensive agents UNIVERSITY OF MIAMI (US) 1982-03-24 EP disclosed