SCHEMBL7278280

SCHEMBL7278280

CCCn1c(N)c(NC(=O)CC23CC4CC(CC(C4)C2)C3)c(=O)n(CCC)c1=O

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
GAA P10253 2/20 0.45
HSD17B10 Q99714 1/20 0.45
CYP2C19 P33261 1/20 0.44
EPHX2 P34913 1/20 0.43
P2RX7 Q99572 5/20 0.43
ADORA1 P30542 1/20 0.42
ALDH1A1 P00352 1/20 0.42
GPR55 Q9Y2T6 1/20 0.40
CA12 O43570 1/20 0.40
CA9 Q16790 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7270332 0.85 DHFR (0.48) SMN1; SMN2ADORA1ALDH1A1
SCHEMBL7279899 0.81 ADORA1 (0.44) GAAP2RX7ADORA1ALDH1A1
SCHEMBL7436318 0.75 ADORA1 (0.46) LMNAGAAHSD17B10ADORA1ALDH1A1
SCHEMBL8705434 0.75 ADORA1 (0.39) GAAADORA1ALDH1A1
SCHEMBL10858163 0.75 ALDH1A1 (0.43) LMNASMN1; SMN2GAAHSD17B10ADORA1
SCHEMBL8706002 0.75 ADORA1 (0.36) LMNAGAAHSD17B10ADORA1ALDH1A1
SCHEMBL8710355 0.73 TDP1 (0.35) LMNAGAAHSD17B10ADORA1ALDH1A1
SCHEMBL8397308 0.73 ADORA2A (0.42) GAAHSD17B10ADORA1ALDH1A1
SCHEMBL7278269 0.72 KCNQ3 (0.46) GAAHSD17B10ALDH1A1
SCHEMBL7274817 0.71 NPSR1 (0.38) LMNASMN1; SMN2GAAHSD17B10CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0415456-B1 Xanthine compounds KYOWA HAKKO KOGYO KK (JP) 1996-06-26 EP disclosed
US-5525607-A DIURETICS, BRONCHODILATORS, RENAL PROTECTING AGENTS KYOWA HAKKO KOGYO CO., LTD (JP) 1996-06-11 US disclosed
US-5290782-A Bronchodilator agents, diuretics for renal protective agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-03-01 US disclosed
EP-0415456-A2 Xanthine compounds KYOWA HAKKO KOGYO CO., LTD. (JP) 1991-03-06 EP disclosed