SCHEMBL8710355

SCHEMBL8710355

CCCn1c(N)c(NC(=O)C23CC4CC2CC(C3)C4=O)c(=O)n(CCC)c1=O

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.35
ADORA1 P30542 9/20 0.35
ADORA2A P29274 3/20 0.35
ADORA3 P0DMS8 2/20 0.35
ADORA2B P29275 1/20 0.35
SLC6A3 Q01959 1/20 0.35
SLC22A6 Q4U2R8 1/20 0.35
SLC22A8 Q8TCC7 1/20 0.35
SLC22A11 Q9NSA0 1/20 0.35
GAA P10253 2/20 0.34
EEF2K O00418 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HSD17B10 Q99714 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8706002 0.85 ADORA1 (0.36) TDP1ADORA1ADORA2AADORA3ADORA2B
SCHEMBL8709010 0.83 KDM4E (0.46) GAAALDH1A1LMNA
SCHEMBL7436318 0.82 ADORA1 (0.46) ADORA1ADORA2AADORA3ADORA2BSLC6A3
SCHEMBL8705434 0.81 ADORA1 (0.39) TDP1ADORA1ADORA2AADORA3ADORA2B
SCHEMBL8707133 0.81 PDE4A (0.38) TDP1ADORA1ADORA2AADORA3ADORA2B
SCHEMBL8397308 0.80 ADORA2A (0.42) ADORA1ADORA2AADORA3ADORA2BSLC6A3
SCHEMBL8208161 0.78 ALDH1A1 (0.40) TDP1ADORA1ADORA2AADORA3ADORA2B
SCHEMBL7279799 0.77 CNR2 (0.40) TDP1ADORA1ADORA2AADORA3ADORA2B
SCHEMBL7269080 0.76 CNR2 (0.39) ADORA1ADORA2AADORA3ADORA2BSLC6A3
SCHEMBL7278280 0.73 LMNA (0.48) ADORA1GAAALDH1A1HSD17B10LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0619316-B1 Xanthine derivatives KYOWA HAKKO KOGYO KK (JP) 1998-08-12 EP disclosed
EP-0619316-A1 Xanthine derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-10-12 EP disclosed