SCHEMBL7278539

SCHEMBL7278539

CC(C)[C@H](N)C(=O)N(C(=O)CCc1ccccc1)[C@@H](C)C(=O)NC(C(C(=O)O)C(C)(C)C)C(O)C(F)(F)CCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.34
MMP2 P08253 11/20 0.33
MMP3 P08254 6/20 0.33
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
HTT P42858 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MMP1 P03956 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275377 0.96 MMP2 (0.35) MLYCDMMP2MMP3KMT2AMEN1
SCHEMBL9153609 0.86 CASP1 (0.37) MLYCDKMT2AMEN1HTTL3MBTL1
SCHEMBL7287140 0.84 CASP1 (0.43) MLYCDMMP2MMP3KMT2AMEN1
SCHEMBL7275911 0.80 CASP1 (0.52) MMP2MMP3MMP1
SCHEMBL7277381 0.75 CASP1 (0.58) MMP2MMP3
SCHEMBL7277260 0.72 CASP1 (0.41) KMT2AMEN1
SCHEMBL7285059 0.72 CASP3 (0.44)
SCHEMBL7277122 0.71 CASP1 (0.51)
SCHEMBL7301728 0.71 CTSC (0.47) KMT2AMEN1
SCHEMBL7286995 0.71 CASP1 (0.40) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0519748-B1 Peptidyl derivatives as inhibitors of interleukin-1B converting enzyme MERCK & CO INC (US) 1998-09-02 EP disclosed
US-5434248-A Peptidyl derivatives as inhibitors of interleukin-1β converting enzyme MERCK & CO., INC. (US) 1995-07-18 US disclosed
EP-0519748-A2 Peptidyl derivatives as inhibitors of interleukin-1B converting enzyme MERCK & CO. INC. (US) 1992-12-23 EP disclosed