SCHEMBL7280204

SCHEMBL7280204

Nc1ccc(CCC(=O)C(N)[C@@H]2C[C@@H](CC(=O)O)C(=O)N2CCCc2ccccc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.39
ALDH1A1 P00352 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MAOB P27338 2/20 0.36
PTGER4 P35408 2/20 0.34
FAAH O00519 5/20 0.33
PTGER3 P43115 1/20 0.33
LTA4H P09960 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275947 0.92 ALDH1A1 (0.37) SIGMAR1ALDH1A1TSHRSMN1; SMN2PTGER4
SCHEMBL7282203 0.89 SIGMAR1 (0.43) SIGMAR1ALDH1A1TSHRSMN1; SMN2PTGER4
SCHEMBL7272761 0.89 SIGMAR1 (0.43) SIGMAR1ALDH1A1TSHRSMN1; SMN2MAOB
SCHEMBL7283910 0.88 SIGMAR1 (0.40) SIGMAR1ALDH1A1TSHRSMN1; SMN2PTGER4
SCHEMBL7272947 0.87 SIGMAR1 (0.40) SIGMAR1ALDH1A1TSHRSMN1; SMN2PTGER4
SCHEMBL7281938 0.87 SIGMAR1 (0.40) SIGMAR1ALDH1A1TSHRSMN1; SMN2PTGER4
SCHEMBL7281748 0.87 SIGMAR1 (0.40) SIGMAR1ALDH1A1TSHRSMN1; SMN2PTGER4
SCHEMBL7276485 0.86 ITGB3 (0.41) ALDH1A1TSHRSMN1; SMN2
SCHEMBL7281960 0.83 ALDH1A1 (0.35) SIGMAR1ALDH1A1TSHRSMN1; SMN2PTGER4
SCHEMBL8943728 0.83 SIGMAR1 (0.40) SIGMAR1MAOBFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0483667-B1 Cyclic imino derivatives, process for their preparation and drugs containing them THOMAE GMBH DR K (DE) 1998-02-04 EP disclosed
US-5591769-A PYRROLIDINE DERIVATIVES; ANTICOAGULANTS KARL THOMAE GMBH (DE) 1997-01-07 US disclosed
EP-0483667-A2 Cyclic imino derivatives, process for their preparation and drugs containing them Dr. Karl Thomae GmbH (DE) 1992-05-06 EP disclosed