SCHEMBL7280800

SCHEMBL7280800

COC(=O)CCc1ccc(N2CCN(c3ccc4c(c3)CC/C4=N/O)C2=O)cc1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.36
HRH3 Q9Y5N1 1/20 0.36
HTT P42858 1/20 0.36
BRAF P15056 4/20 0.35
PTPN1 P18031 4/20 0.35
S1PR1 P21453 1/20 0.35
ROCK2 O75116 1/20 0.35
P2RX3 P56373 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7280804 1.00 HDAC1 (0.36) HDAC1HRH3HTTBRAFPTPN1
SCHEMBL7393684 0.94 HRH3 (0.37) HDAC1HRH3BRAFPTPN1S1PR1
SCHEMBL7284346 0.88 HDAC1 (0.39) HDAC1HRH3PTPN1S1PR1ROCK2
SCHEMBL7390094 0.84 BAZ2B (0.40) HRH3
SCHEMBL8559518 0.80 HRH3 (0.41) HDAC1HRH3S1PR1POLB
Hydrochloric Acid SCHEMBL8564996 0.79 HRH3 (0.40) HDAC1HRH3S1PR1POLB
SCHEMBL8559578 0.78 HTR6 (0.42) HDAC1HRH3S1PR1POLB
Hydrochloric Acid SCHEMBL8566255 0.78 HTR6 (0.41) HDAC1HRH3S1PR1POLB
SCHEMBL8563370 0.77 ASIC3 (0.40) HDAC1HRH3S1PR1ROCK2
SCHEMBL27397736 0.77 MEN1 (0.51) HDAC1HRH3PTPN1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650424-A ANTIAGGLOMERANTS USING IMIDAZOLIDINDIONES DR. KARL THOMAE GMBH (DE) 1997-07-22 US disclosed
EP-0503548-B1 Cyclic urea derivatives, medicaments contaning them and process for their preparation THOMAE GMBH DR K (DE) 1997-06-04 EP disclosed
US-5478942-A Antiinflammatory agents, antiagglomerants KARL THOMAE GMBH (DE) 1995-12-26 US disclosed
US-5276049-A Treatment of thrombosis DR. KARL THOMAE GMBH (DE) 1994-01-04 US disclosed
EP-0503548-A1 Cyclic urea derivatives, medicaments contaning them and process for their preparation Dr. Karl Thomae GmbH (DE) 1992-09-16 EP disclosed