SCHEMBL7280865

SCHEMBL7280865

COc1cc(N(C)C)ccc1[C]=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.43
HSD17B10 Q99714 3/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
HPGD P15428 2/20 0.43
KDM4E B2RXH2 1/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
LMNA P02545 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CYP3A4 P08684 2/20 0.42
TSHR P16473 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2C19 P33261 1/20 0.42
NQO2 P16083 1/20 0.41
TUBB1 Q9H4B7 2/20 0.40
TUBB4A P04350 1/20 0.40
TUBB P07437 1/20 0.40
TUBA3C P0DPH7 1/20 0.40
TUBA1B P68363 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4308489 0.81 AR (0.50) ALDH1A1KDM4EGAAUSP2PGR
SCHEMBL11619380 0.81 ELANE (0.40) ALDH1A1HSD17B10HPGDKDM4EGAA
SCHEMBL96290 0.79 CA12 (0.56) ALDH1A1HPGDMEN1KMT2ACYP3A4
SCHEMBL1107760 0.76 NQO2 (0.63) ALDH1A1HSD17B10SMN1; SMN2HPGDKDM4E
SCHEMBL11593518 0.75 ALDH1A1 (0.39) ALDH1A1HPGDKDM4ECYP3A4USP2
SCHEMBL7671557 0.75 ALDH1A1 (0.40) ALDH1A1HSD17B10SMN1; SMN2HPGDKDM4E
SCHEMBL6210428 0.75 ACHE (0.56) ALDH1A1HPGDKDM4EGAAMEN1
SCHEMBL11309184 0.74 ALDH1A1 (0.44) ALDH1A1HSD17B10SMN1; SMN2HPGDKDM4E
SCHEMBL4392239 0.73 TRPV4 (0.50) ALDH1A1HPGDKDM4ELMNAMEN1
SCHEMBL7242037 0.73 ALDH1A1 (0.56) ALDH1A1HSD17B10SMN1; SMN2HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470514-B1 Carbostyril derivatives and pharmaceutical composition containing the same OTSUKA PHARMA CO LTD (JP) 1997-02-19 EP disclosed
US-5300513-A Vasopressin antagonists; vasodilators, hypotensive agents, water diuretics, and platelet agglutination inhibitors OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-05 US disclosed
EP-0470514-A1 Carbostyril derivatives and pharmaceutical composition containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-02-12 EP disclosed