SCHEMBL72819

SCHEMBL72819

CCOC(=O)Cc1cc(Cl)c(NC(=O)c2coc3ccccc23)cc1F

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOB P27338 13/20 0.45
MAPT P10636 2/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
CA5A P35218 2/20 0.43
CA7 P43166 2/20 0.43
CA5B Q9Y2D0 2/20 0.43
GAA P10253 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ITGB1 P05556 4/20 0.41
ITGA4 P13612 4/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL73880 0.91 MAOB (0.47) MAOBMAPTNPC1RAB9ACA12
SCHEMBL70950 0.86 MAOB (0.50) MAOBMAPTNPC1RAB9ACA12
SCHEMBL91531 0.82 MAOB (0.54) MAOBMAPTNPC1RAB9ACA12
SCHEMBL72217 0.81 MAPT (0.41) MAOBMAPTNPC1RAB9AGAA
SCHEMBL72295 0.81 PKM (0.54) MAPTNPC1SMN1; SMN2ITGB1ITGA4
SCHEMBL14592698 0.77 ITGB1 (0.56) NPC1RAB9AGAASMN1; SMN2ITGB1
SCHEMBL14592356 0.77 SMN1; SMN2 (0.44) NPC1RAB9ASMN1; SMN2ITGB1ITGA4
SCHEMBL14491705 0.77 ITGB1 (0.55) MAPTNPC1RAB9AGAASMN1; SMN2
SCHEMBL72182 0.77 MAOB (0.53) MAOBMAPTNPC1RAB9ACA12
SCHEMBL91556 0.76 MAOB (0.57) MAOBMAPTNPC1RAB9ACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1961750-B1 VLA-4 INHIBITORY DRUG DAIICHI SANKYO CO LTD (JP) 2013-09-18 EP disclosed