SCHEMBL72295

SCHEMBL72295

CCOC(=O)Cc1cc(Cl)c(NC(=O)c2c[nH]c3ccccc23)cc1F

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.54
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
NPC1 O15118 2/20 0.47
NHERF1 O14745 1/20 0.46
CFTR P13569 3/20 0.46
TDP1 Q9NUW8 1/20 0.44
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C19 P33261 2/20 0.44
MAPT P10636 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
ITGB1 P05556 1/20 0.42
ITGA4 P13612 1/20 0.42
LMNA P02545 2/20 0.42
ALDH1A1 P00352 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL71626 0.91 PKM (0.57) PKMMEN1KMT2ANPC1NHERF1
SCHEMBL73753 0.86 NHERF1 (0.51) MEN1KMT2ANPC1NHERF1CFTR
SCHEMBL2438042 0.83 ITGB1 (0.53) PKMMEN1KMT2ANPC1NHERF1
SCHEMBL5708329 0.82 PKM (0.40) PKMKMT2ANHERF1ALDH1A1KDM4E
SCHEMBL14592698 0.82 ITGB1 (0.56) PKMKMT2ANPC1SMN1; SMN2ITGB1
SCHEMBL92571 0.82 NPC1 (0.57) MEN1KMT2ANPC1NHERF1CFTR
SCHEMBL72819 0.81 MAOB (0.45) NPC1MAPTSMN1; SMN2ITGB1ITGA4
SCHEMBL72217 0.81 MAPT (0.41) MEN1KMT2ANPC1CYP1A2CYP3A4
SCHEMBL14491705 0.77 ITGB1 (0.55) MEN1KMT2ANPC1TDP1MAPT
SCHEMBL14592356 0.77 SMN1; SMN2 (0.44) MEN1KMT2ANPC1CYP1A2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1961750-B1 VLA-4 INHIBITORY DRUG DAIICHI SANKYO CO LTD (JP) 2013-09-18 EP disclosed