SCHEMBL7282298

SCHEMBL7282298

N#CC(C=O)c1cc(Cl)cc(Cl)c1Cl.[NaH]

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.37
AHR P35869 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
ERN1 O75460 1/20 0.31
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5070145 0.98 ALDH1A1 (0.38) ALDH1A1AHRHPGDTSHRHSD17B10
SCHEMBL7282307 0.97 ALDH1A1 (0.37) ALDH1A1AHRHPGDTSHRHSD17B10
SCHEMBL5069257 0.77 ALDH1A1 (0.45) ALDH1A1MAPT
SCHEMBL6049601 0.74 PNMT (0.43) ALDH1A1TSHR
SCHEMBL8894567 0.74
SCHEMBL8897584 0.72
SCHEMBL7273201 0.72 ERN1 (0.34) TSHRERN1
SCHEMBL16093967 0.68 KDM4E (0.43) ALDH1A1HPGDERN1
SCHEMBL5073554 0.68 ALDH1A1 (0.35) ALDH1A1AHRHPGDTSHRHSD17B10
SCHEMBL11788286 0.66 GABRA1 (0.37) ALDH1A1AHRHPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0372934-B1 Pharmacologically active CNS compounds WELLCOME FOUND (GB) 1996-10-23 EP disclosed
EP-0459819-B1 Pharmacologically active CNS compound WELLCOME FOUND (GB) 1996-08-14 EP disclosed
CN-1117046-A Method for preparing pharmaceutically active CNS compounds WELLCOME FOUND (GB) 1996-02-21 CN disclosed
CN-1113487-A Method for preparing pharmaceutically active CNS compounds WELLCOME FOUND (GB) 1995-12-20 CN disclosed
EP-0679645-A1 Pharmacologically active CNS pyridmidin compounds THE WELLCOME FOUNDATION LIMITED (GB) 1995-11-02 EP disclosed
EP-0459819-A2 Pharmacologically active CNS compound THE WELLCOME FOUNDATION LIMITED (GB) 1991-12-04 EP disclosed
CN-1052306-A Compounds having pharmacological activity on the central nervous system WELLCOME FOUND (GB) 1991-06-19 CN disclosed