SCHEMBL7283452

SCHEMBL7283452

CS(=O)(=O)C[C@H](NC(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.54
CTSS P25774 3/20 0.53
CTSL P07711 2/20 0.53
CTSB P07858 2/20 0.53
CASP1 P29466 3/20 0.53
ALDH1A1 P00352 1/20 0.52
ALOX15 P16050 1/20 0.52
MMP13 P45452 3/20 0.52
PPARA Q07869 2/20 0.52
PPARG P37231 1/20 0.52
TACR1 P25103 2/20 0.51
KYNU Q16719 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22783671 0.87 PPARA (0.53) CTSKCTSSCTSLCTSBCASP1
SCHEMBL2749553 0.86 PPARA (0.53) CTSKCTSSCTSLCTSBCASP1
SCHEMBL9686663 0.86 CA12 (0.57) CTSKCTSSCTSLCTSBCASP1
SCHEMBL7349434 0.86 CA12 (0.57) CTSKCTSSCTSLCTSBCASP1
SCHEMBL12226071 0.85 MMP13 (0.51) CTSKCTSSCTSLCTSBCASP1
SCHEMBL3805426 0.84 CA2 (0.55) CTSKCTSSCTSLCTSB
SCHEMBL457686 0.84 PPARA (0.57) CTSKCTSSCTSLCTSBCASP1
SCHEMBL201710 0.84 PPARA (0.57) CTSKCTSSCTSLCTSBCASP1
SCHEMBL295865 0.84 PPARA (0.57) CTSKCTSSCTSLCTSBCASP1
SCHEMBL4972916 0.84 CTSK (0.52) CTSKCTSSCTSLCTSBCASP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696134-A Irreversible HIV protease inhibitors, intermediates, compositions and processes for the preparation thereof LG CHEMICAL LIMITED (KR) 1997-12-09 US disclosed
EP-0687675-A2 Irreversible HIV protease inhibitors, intermediates, compositions and processes for the preparation thereof LG Chemical Limited (KR) 1995-12-20 EP disclosed