SCHEMBL7283889

SCHEMBL7283889

CC(CNc1ncc(-c2ccncc2)cc1C#N)OC(=O)c1cccnc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
ALDH1A1 P00352 4/20 0.41
MAPT P10636 1/20 0.41
CFTR P13569 2/20 0.40
GAK O14976 1/20 0.39
STK16 O75716 1/20 0.39
PIM1 P11309 1/20 0.39
AXL P30530 1/20 0.39
NEK2 P51955 1/20 0.39
STK3 Q13188 1/20 0.39
STK11 Q15831 1/20 0.39
AAK1 Q2M2I8 1/20 0.39
BMP2K Q9NSY1 1/20 0.39
TNIK Q9UKE5 1/20 0.39
KMT2A Q03164 5/20 0.38
MEN1 O00255 3/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7292041 0.83 KDM4E (0.51) LMNACYP1A2CYP3A4ALDH1A1MAPT
SCHEMBL4591354 0.79 CFTR (0.59) LMNACYP1A2CYP3A4CFTRGAK
Water SCHEMBL7302779 0.79 CFTR (0.59) LMNACYP1A2CYP3A4CFTRGAK
SCHEMBL7284179 0.78 GLA (0.42) CYP1A2ALDH1A1AAK1BMP2KRAB9A
Hydrochloric Acid SCHEMBL7298103 0.77 ALDH1A1 (0.48) LMNACYP1A2CYP3A4ALDH1A1MAPT
SCHEMBL7292620 0.77 KDM4E (0.50) LMNACYP1A2CYP3A4ALDH1A1MAPT
SCHEMBL7283041 0.75 CLK4 (0.39) CYP3A4ALDH1A1AXLAAK1KMT2A
SCHEMBL7282598 0.75 KDM4E (0.44) LMNACYP1A2CYP3A4ALDH1A1MAPT
SCHEMBL7284472 0.73 L3MBTL1 (0.51) LMNACYP1A2CYP3A4ALDH1A1MAPT
SCHEMBL11238008 0.73 GSK3A (0.45) LMNACYP1A2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0200024-B1 3-CYANO-PYRIDINES, PROCESS FOR THEIR PREPARATION AND THEIR PHARMACEUTICAL USE ARZNEIMITTELWERK DRESDEN GmbH (DE) 1992-07-01 EP disclosed
EP-0200024-A2 3-Cyano-pyridines, process for their preparation and their pharmaceutical use ARZNEIMITTELWERK DRESDEN GmbH (DE) 1986-11-05 EP disclosed