SCHEMBL7285483

SCHEMBL7285483

CC(C)(C)OC(=O)N1CCc2ccc(C(=O)NC[C@@H]3C[C@@H](CC(=O)O)C(=O)N3CCCc3ccccc3)cc2C1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.41
KDM4E B2RXH2 1/20 0.41
PKM P14618 1/20 0.41
ESR2 Q92731 1/20 0.38
SIGMAR1 Q99720 4/20 0.37
PRMT5 O14744 1/20 0.37
ITGB3 P05106 2/20 0.37
ITGA2B P08514 2/20 0.37
TMEM97 Q5BJF2 1/20 0.36
HTR1A P08908 2/20 0.36
NAMPT P43490 3/20 0.36
PTPN1 P18031 1/20 0.36
P2RX3 P56373 1/20 0.36
OPRM1 P35372 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7286501 0.96 KDM4E (0.43) NR1H2KDM4EPKMESR2SIGMAR1
SCHEMBL7283192 0.94 NR1H2 (0.40) NR1H2KDM4EPKMESR2SIGMAR1
SCHEMBL7277905 0.94 KDM4E (0.41) KDM4EPKMSIGMAR1ITGB3ITGA2B
SCHEMBL7285724 0.93 ITGB3 (0.41) NR1H2KDM4EPKMESR2SIGMAR1
SCHEMBL7275338 0.89 ITGB3 (0.40) NR1H2KDM4EPKMSIGMAR1ITGB3
SCHEMBL7276445 0.88 NAMPT (0.40) KDM4EPKMSIGMAR1HTR1ANAMPT
SCHEMBL7286896 0.88 NAMPT (0.39) NR1H2KDM4EPKMESR2SIGMAR1
SCHEMBL7277666 0.88 TMPRSS2 (0.41) ITGB3ITGA2BHTR1ANAMPT
SCHEMBL7283282 0.87 KDM4E (0.41) NR1H2KDM4EPKMESR2SIGMAR1
SCHEMBL7286536 0.87 ITGB3 (0.43) NR1H2KDM4EPKMSIGMAR1ITGB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed