SCHEMBL7286501

SCHEMBL7286501

CC(C)(C)OC(=O)N1CCc2ccc(C(=O)NC[C@@H]3C[C@@H](CC(=O)O)C(=O)N3CCCc3ccccc3)cc2CC1

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
PKM P14618 1/20 0.43
SIGMAR1 Q99720 3/20 0.38
HTR1A P08908 2/20 0.37
MAPK14 Q16539 1/20 0.37
ESR2 Q92731 1/20 0.36
STS P08842 1/20 0.36
NR1H2 P55055 1/20 0.36
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
MTNR1A P48039 1/20 0.35
GPR119 Q8TDV5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7285483 0.96 NR1H2 (0.41) KDM4EPKMSIGMAR1HTR1AESR2
SCHEMBL7275338 0.93 ITGB3 (0.40) KDM4EPKMSIGMAR1MAPK14NR1H2
SCHEMBL7277905 0.92 KDM4E (0.41) KDM4EPKMSIGMAR1HTR1AITGB3
SCHEMBL7283282 0.91 KDM4E (0.41) KDM4EPKMSIGMAR1HTR1AMAPK14
SCHEMBL7283192 0.91 NR1H2 (0.40) KDM4EPKMSIGMAR1HTR1AESR2
SCHEMBL7285724 0.89 ITGB3 (0.41) KDM4EPKMSIGMAR1MAPK14ESR2
SCHEMBL9251785 0.87 TMPRSS2 (0.41) HTR1AITGB3ITGA2B
SCHEMBL7275263 0.87 TMPRSS2 (0.41) HTR1AITGB3ITGA2B
SCHEMBL7276445 0.86 NAMPT (0.40) KDM4EPKMSIGMAR1HTR1A
SCHEMBL7288079 0.86 KDM4E (0.49) KDM4EPKMSIGMAR1STSSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed