SCHEMBL7285571

SCHEMBL7285571

N[C@H](Cc1ccccc1)C(=O)N1CCN(CC(=O)OCc2ccccc2)C(=O)C1

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 6/20 0.52
SLC15A1 P46059 1/20 0.46
OPRD1 P41143 2/20 0.44
AKT1 P31749 3/20 0.43
PLAU P00749 1/20 0.43
PLAUR Q03405 1/20 0.43
AKT2 P31751 1/20 0.43
AKT3 Q9Y243 1/20 0.43
DPP4 P27487 5/20 0.42
DPP7 Q9UHL4 3/20 0.42
DPP8 Q6V1X1 2/20 0.42
ROCK2 O75116 1/20 0.40
CYP3A4 P08684 1/20 0.40
FAP Q12884 1/20 0.40
DPP9 Q86TI2 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7285561 0.99 HDAC8 (0.54) HDAC8SLC15A1OPRD1AKT1PLAU
SCHEMBL7276024 0.83 ITGB3 (0.43) DPP4
Hydrochloric Acid SCHEMBL7278971 0.82 ITGB3 (0.43) DPP4
SCHEMBL16465214 0.78 HDAC8 (0.58) HDAC8SLC15A1OPRD1AKT1PLAU
SCHEMBL16466269 0.78 HDAC8 (0.58) HDAC8SLC15A1OPRD1AKT1PLAU
SCHEMBL28018784 0.78 HDAC8 (0.58) HDAC8SLC15A1OPRD1AKT1PLAU
SCHEMBL25426510 0.78 ALDH1A1 (0.54)
SCHEMBL29218649 0.77 ALDH1A1 (0.45)
SCHEMBL7368700 0.77 RAB9A (0.48)
SCHEMBL23291427 0.76 PRMT5 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0529858-B1 2-Piperazinone compounds, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-15 EP disclosed
US-5294713-A Inhibiting cell adhesion TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-03-15 US disclosed
EP-0529858-A1 2-Piperazinone compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1993-03-03 EP disclosed