SCHEMBL7286164

SCHEMBL7286164

Cc1ccccc1S(=O)(=O)N[C@@H](CCCCN)C(=O)C(=O)CCl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.50
MMP9 P14780 1/20 0.50
ITGAV P06756 3/20 0.46
SLC1A3 P43003 1/20 0.44
SLC1A2 P43004 1/20 0.44
SLC1A1 P43005 1/20 0.44
ITGA2 P17301 1/20 0.41
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CASP1 P29466 1/20 0.39
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
BDKRB1 P46663 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
BMP1 P13497 1/20 0.37
ITGB3 P05106 1/20 0.37
PYGL P06737 1/20 0.36
F2 P00734 2/20 0.36
TBXAS1 P24557 1/20 0.36
KAT6A Q92794 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27465967 1.00 MMP2 (0.50) MMP2MMP9ITGAVSLC1A3SLC1A2
SCHEMBL28658079 0.88 MMP2 (0.49) MMP2MMP9ITGAVSLC1A3SLC1A2
Hydrochloric Acid SCHEMBL29175312 0.87 MMP2 (0.48) MMP2MMP9ITGAVSLC1A3SLC1A2
SCHEMBL457771 0.84 MMP9 (0.65) MMP2MMP9ITGAVSLC1A3SLC1A2
SCHEMBL27737068 0.83 MMP9 (0.60) MMP2MMP9ITGAVSLC1A3SLC1A2
SCHEMBL1305743 0.82 MMP2 (0.56) MMP2MMP9SLC1A3SLC1A2SLC1A1
SCHEMBL1305745 0.82 MMP2 (0.56) MMP2MMP9SLC1A3SLC1A2SLC1A1
SCHEMBL11207292 0.82 RECQL (0.52) MMP2MMP9ITGAVSLC1A3SLC1A2
Hydrochloric Acid SCHEMBL28193637 0.82 MMP2 (0.59) MMP2MMP9ITGAVSLC1A3SLC1A2
SCHEMBL1469951 0.80 POLB (0.52) MMP2MMP9ITGAVSLC1A3SLC1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0263903-A1 Method for preparing specific inhibitors of virus-specified proteases E.I. DU PONT DE NEMOURS AND COMPANY (US) 1988-04-20 EP disclosed
EP-0263214-A1 Tetrapeptide methyl ketone inhibitors of viral proteases E.I. DU PONT DE NEMOURS AND COMPANY (US) 1988-04-13 EP disclosed
EP-0263202-A1 Inhibition of viral protease activity by peptide halomethyl ketones E.I. DU PONT DE NEMOURS AND COMPANY (US) 1988-04-13 EP disclosed
US-4652552-A ENZYME INHIBITORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-03-24 US disclosed
US-4644055-A HALOMETHYL KETONE OR METHYL KETONE COVALENTLY LINKED TO PEPTIDE SEQUENCE E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-02-17 US disclosed
US-4636492-A ENZYME INHIBITORS E. I. DU PONT DE NEMOURS AND COMPANY (US) 1987-01-13 US disclosed