SCHEMBL7286567

SCHEMBL7286567

COC(=O)C[C@@H]1C[C@@H](COc2ccc(-c3ccc(C#N)cc3)cc2)N(C(=O)c2cccnc2)C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
KCNA5 P22460 1/20 0.39
PORCN Q9H237 1/20 0.39
FNTA P49354 1/20 0.38
FNTB P49356 1/20 0.38
PIK3CD O00329 1/20 0.38
GAK O14976 1/20 0.38
STK16 O75716 1/20 0.38
PIM1 P11309 1/20 0.38
AXL P30530 1/20 0.38
NEK2 P51955 1/20 0.38
STK3 Q13188 1/20 0.38
STK11 Q15831 1/20 0.38
AAK1 Q2M2I8 1/20 0.38
BMP2K Q9NSY1 1/20 0.38
TNIK Q9UKE5 1/20 0.38
CHRNA7 P36544 2/20 0.38
KCNH2 Q12809 1/20 0.37
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7283484 0.89 KCNA5 (0.42) KCNA5ALDH1A1
Hydrochloric Acid SCHEMBL7284136 0.88 ITGB3 (0.39) PIK3CDKCNH2ALDH1A1
Hydrochloric Acid SCHEMBL7277269 0.85 PIK3CD (0.35) PIK3CDCHRNA7KCNH2ALDH1A1
Hydrochloric Acid SCHEMBL7277857 0.83 AOC3 (0.36) PIK3CDKCNH2ALDH1A1
SCHEMBL7272380 0.83 MMP2 (0.41) CHRNA7ALDH1A1
SCHEMBL7275606 0.82 MMP2 (0.42) CHRNA7ALDH1A1
SCHEMBL7272704 0.80 POLB (0.39) CHRNA7ALDH1A1
SCHEMBL7283917 0.79 SLC6A7 (0.40) CHRNA7SCN9A
SCHEMBL7275597 0.79 KDM4E (0.40) CHRNA7
SCHEMBL7274649 0.79 CHRNA7 (0.43) CHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0528369-B1 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation BOEHRINGER INGELHEIM PHARMA (DE) 1999-11-24 EP disclosed
US-5455348-A Anticoagulants Thomae, Karl (DE) 1995-10-03 US disclosed
EP-0528369-A2 Cyclic imino derivatives, pharmaceutical compositions containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-02-24 EP disclosed