SCHEMBL7287387

SCHEMBL7287387

O=C1CC2CCSc3ccccc3C2=NN1c1ccc(Br)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.34
CES2 O00748 2/20 0.34
ACHE P22303 2/20 0.34
ALDH1A1 P00352 2/20 0.33
RECQL P46063 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
EP300 Q09472 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
MEN1 O00255 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
KMT2A Q03164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7294604 0.91 PDE4A (0.39) GAACES2ACHEALDH1A1RECQL
SCHEMBL7292065 0.90 HTT (0.37) GAACES2ACHEALDH1A1SMN1; SMN2
SCHEMBL7291459 0.90 CNR2 (0.36) CES2ACHESMN1; SMN2PDE4APDE4B
SCHEMBL10569584 0.89 KDM4E (0.38) ALDH1A1RECQLPDE4APDE4BPDE4C
SCHEMBL7289330 0.89 MIF (0.34) ACHEPDE4APDE4BPDE4CPDE4D
SCHEMBL7286210 0.89 GABRP (0.41) ACHEALDH1A1SMN1; SMN2PDE4APDE4B
SCHEMBL10561260 0.88 ACHE (0.36) GAACES2ACHEALDH1A1RECQL
SCHEMBL7286216 0.86 IDO1 (0.34) PDE4APDE4BPDE4CPDE4DMAPT
SCHEMBL7290542 0.86 MAPT (0.41) GAACES2ACHEALDH1A1SMN1; SMN2
SCHEMBL10570971 0.85 MAPT (0.45) GAAALDH1A1SMN1; SMN2MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281045-B1 BENZOTHIEPINO (5,4-C) PYRIDAZINE COMPOUNDS AND THEIR PHARMACEUTICAL USES Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1991-12-27 EP claimed
EP-0281045-A1 Benzothiepino (5,4-c) pyridazine compounds and their pharmaceutical uses Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1988-09-07 EP disclosed