SCHEMBL7288371

SCHEMBL7288371

N=C(N)N(CCCc1c[nH]cn1)CCN(Cc1cccs1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 4/20 0.35
ADRA2B P18089 3/20 0.35
CHRM2 P08172 3/20 0.35
CHRM1 P11229 3/20 0.35
CYP2D6 P10635 2/20 0.35
DRD1 P21728 2/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
OPRM1 P35372 2/20 0.35
SLC6A3 Q01959 2/20 0.35
KCNH2 Q12809 2/20 0.35
CYP1A2 P05177 1/20 0.35
CHRM5 P08912 1/20 0.35
CYP2C9 P11712 1/20 0.35
NFKB1 P19838 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HRH1 P35367 1/20 0.35
HTR2B P41595 1/20 0.35
HTR6 P50406 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9828576 0.86 HRH4 (0.39) ADRA2ACYP2D6OPRM1SLC6A3KCNH2
Hydrochloric Acid SCHEMBL9827176 0.85 GRIN2D (0.40) ADRA2ACYP2D6OPRM1SLC6A3KCNH2
SCHEMBL7288663 0.81 SCN5A (0.34) ADRA2AADRA2BCHRM2CHRM1CYP2D6
SCHEMBL9828326 0.80 HRH4 (0.33) KCNH2ALDH1A1
SCHEMBL9828851 0.80 GBA1 (0.38) CYP2D6CYP1A2TSHRPKMSMN1; SMN2
Hydrochloric Acid SCHEMBL9827568 0.79 GRIN2D (0.33) KCNH2ALDH1A1
SCHEMBL7288384 0.79 SCN5A (0.34) ADRA2AADRA2BADRA2C
Hydrochloric Acid SCHEMBL9827508 0.79 GRIN2D (0.36) CYP2D6KCNH2TSHRALDH1A1SMN1; SMN2
SCHEMBL9828412 0.76 CHRM2 (0.46) ADRA2AADRA2BCHRM2CHRM1CYP2D6
Hydrochloric Acid SCHEMBL9827919 0.75 LMNA (0.47) ADRA2AADRA2BCHRM2CHRM1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0262448-B1 IMIDAZOLYLGUANIDINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM HEUMANN PHARMA GMBH & CO (DE) 1991-12-18 EP disclosed