SCHEMBL7288409

SCHEMBL7288409

[CH]1CNCCC1CCCCCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.40
GBA1 P04062 1/20 0.40
SIGMAR1 Q99720 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27644564 0.98 GBA1 (0.41) CYP19A1GBA1SIGMAR1
SCHEMBL2089535 0.80 ITGB3 (0.40) SIGMAR1
SCHEMBL11537058 0.78 GBA1 (0.58) GBA1SIGMAR1
SCHEMBL27525435 0.77 GBA1 (0.56) GBA1SIGMAR1
SCHEMBL9820951 0.76 CYP19A1 (0.40) CYP19A1SIGMAR1
SCHEMBL7297794 0.76 CYP19A1 (0.40) CYP19A1SIGMAR1
SCHEMBL3358034 0.76 GBA1 (0.59) GBA1SIGMAR1
SCHEMBL29139845 0.72 SIGMAR1 (0.47) SIGMAR1
SCHEMBL82734 0.70 GBA1 (0.61) GBA1SIGMAR1
SCHEMBL9820891 0.70 CYP19A1 (0.40) CYP19A1GBA1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652247-A VASOPRESSIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD (JP) 1997-07-29 US disclosed
US-5436254-A Vaopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1995-07-25 US disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
EP-0382185-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1994-06-15 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
US-5225402-A Vasopressin antagonist, vasodilation, hypotensive, diuretics and anticoagulants OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-06 US disclosed
EP-0382185-A2 Carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-08-16 EP disclosed