SCHEMBL7288684

SCHEMBL7288684

Brc1[c]c2ccccc2[nH]1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
HSD17B10 Q99714 2/20 0.35
GPR3 P46089 1/20 0.35
KDM4E B2RXH2 2/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2A Q12879 1/20 0.33
GRIN2B Q13224 1/20 0.33
GRIN2C Q14957 1/20 0.33
GRIN3A Q8TCU5 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33
PSMB8 P28062 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CA1 P00915 2/20 0.32
CA4 P22748 2/20 0.32
CA6 P23280 2/20 0.32
CA12 O43570 1/20 0.32
CA3 P07451 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11785225 0.75 ALDH1A1 (0.38) ALDH1A1HSD17B10GPR3KDM4EGRIN2D
SCHEMBL29547 0.71 AHR (0.37) ALDH1A1HSD17B10GPR3KDM4EGRIN2D
SCHEMBL4466423 0.71 ALDH1A1 (0.35) ALDH1A1HSD17B10GPR3KDM4EGRIN2D
SCHEMBL2230518 0.71 ALDH1A1 (0.35) ALDH1A1HSD17B10GPR3KDM4EGRIN2D
SCHEMBL8588800 0.71 ALDH1A1 (0.40) ALDH1A1HSD17B10GPR3KDM4EGRIN2D
SCHEMBL5067720 0.71 ALDH1A1 (0.40) ALDH1A1MAPTTDP1HTTSMN1; SMN2
SCHEMBL28824470 0.70 AHR (0.35) ALDH1A1HSD17B10GPR3KDM4EGRIN2D
SCHEMBL7620124 0.69 LMNA (0.33) ALDH1A1MAPTHTR2AHTR2CLMNA
SCHEMBL1972818 0.68 NPC1 (0.41) ALDH1A1HSD17B10GPR3KDM4EGRIN2D
SCHEMBL10813818 0.68 ALDH1A1 (0.32) ALDH1A1HSD17B10GPR3KDM4EGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111533767-A Tetradentate phosphine ligand and preparation method thereof, hydroformylation catalyst and reaction method, and preparation method of 1, 3-propylene glycol 卢海元 2020-08-14 CN claimed
US-4870087-A Indole containing, 2-thienyl-1,2,3,6-tetrahydropyridyls and their pharmaceutical use MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1989-09-26 US claimed
US-4617309-A Sulfur-containing indole derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1986-10-14 US claimed
CN-111533767-A Tetradentate phosphine ligand and preparation method thereof, hydroformylation catalyst and reaction method, and preparation method of 1, 3-propylene glycol 卢海元 2020-08-14 CN disclosed
US-4870087-A Indole containing, 2-thienyl-1,2,3,6-tetrahydropyridyls and their pharmaceutical use MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1989-09-26 US disclosed
EP-0121716-B1 INDOLE DERIVATIVES MERCK PATENT GmbH (DE) 1987-12-09 EP disclosed
US-4617309-A Sulfur-containing indole derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1986-10-14 US disclosed
EP-0105397-B1 SULPHURIC INDOLE DERIVATIVES MERCK PATENT GmbH (DE) 1986-07-16 EP disclosed
EP-0121716-A1 Indole derivatives MERCK PATENT GmbH (DE) 1984-10-17 EP disclosed
EP-0114603-A1 Indole derivatives MERCK PATENT GmbH (DE) 1984-08-01 EP disclosed
EP-0105397-A1 Sulphuric indole derivatives MERCK PATENT GmbH (DE) 1984-04-18 EP disclosed