SCHEMBL7288776

SCHEMBL7288776

Cc1cc(C)c(NC(=O)CN2CCNCC2)c(C)c1

nearest known ligand 0.74

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.74
MEN1 O00255 1/20 0.74
KMT2A Q03164 1/20 0.74
ALOX15 P16050 1/20 0.72
TSHR P16473 3/20 0.57
RAB9A P51151 2/20 0.57
NPC1 O15118 1/20 0.57
TP53 P04637 1/20 0.55
LMNA P02545 2/20 0.50
HTT P42858 1/20 0.49
CHRM5 P08912 1/20 0.49
CHRM3 P20309 1/20 0.49
ALDH1A1 P00352 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1777934 0.85 ALDH1A1 (0.57) POLBMEN1KMT2AALOX15TSHR
SCHEMBL27935848 0.84 MEN1 (0.61) POLBMEN1KMT2AALOX15RAB9A
SCHEMBL9032081 0.83 MEN1 (0.52) POLBMEN1KMT2AALOX15TSHR
Hydrochloric Acid SCHEMBL8554173 0.83 ALDH1A1 (0.55) POLBMEN1KMT2AALOX15TSHR
SCHEMBL7438110 0.82 POLB (0.74) POLBMEN1KMT2AALOX15TSHR
Water SCHEMBL9367224 0.79 MEN1 (0.48) POLBMEN1KMT2AALOX15TSHR
SCHEMBL7278718 0.79 ALDH1A1 (0.62) POLBMEN1KMT2ATSHRNPC1
SCHEMBL9031774 0.78 ALDH1A1 (0.53) POLBMEN1KMT2AALOX15TSHR
SCHEMBL7705614 0.78 POLB (0.55) POLBMEN1KMT2AALOX15TSHR
SCHEMBL1778375 0.77 ALDH1A1 (0.49) POLBMEN1KMT2AALOX15TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4567264-A ADRENERGIC BLOCKING AGENTS SYNTEX (U.S.A.) INC. (US) 1986-01-28 US disclosed
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed
EP-0126449-A1 Cardioselective aryloxy- and arylthio-hydroxypropyl piperazinyl acetanilides wich affect calcium entry SYNTEX (U.S.A.) INC. (US) 1984-11-28 EP disclosed