SCHEMBL7289645

SCHEMBL7289645

O=C1CC2CCSc3ccccc3C2=NN1c1ccc(Cl)c(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KMT2A Q03164 3/20 0.34
MEN1 O00255 2/20 0.34
ADAM17 P78536 1/20 0.34
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34
GRM5 P41594 4/20 0.33
MAPT P10636 2/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
PSMD14 O00487 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10561166 0.89 GAA (0.36) GAAALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL7288071 0.88 KMT2A (0.43) GAAALDH1A1SMN1; SMN2KMT2AMEN1
SCHEMBL7286210 0.88 GABRP (0.41) ALDH1A1CYP2C9CYP2C19SMN1; SMN2KMT2A
SCHEMBL7294604 0.85 PDE4A (0.39) GAAALDH1A1CYP1A2SMN1; SMN2KMT2A
SCHEMBL7292065 0.84 HTT (0.37) GAAALDH1A1CYP1A2SMN1; SMN2KMT2A
SCHEMBL7291459 0.84 CNR2 (0.36) SMN1; SMN2GRM5MAPTTSHR
SCHEMBL7289330 0.84 MIF (0.34) POLB
SCHEMBL7287387 0.84 GAA (0.34) GAAALDH1A1CYP1A2CYP2C9CYP2C19
SCHEMBL10569584 0.84 KDM4E (0.38) ALDH1A1KMT2AMEN1MAPT
SCHEMBL7291194 0.84 ADRA1D (0.34) GAAALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0281045-B1 BENZOTHIEPINO (5,4-C) PYRIDAZINE COMPOUNDS AND THEIR PHARMACEUTICAL USES Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1991-12-27 EP disclosed
US-4849421-A SIDE EFFECT REDUCTION YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1989-07-18 US disclosed
EP-0281045-A1 Benzothiepino (5,4-c) pyridazine compounds and their pharmaceutical uses Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1988-09-07 EP disclosed