SCHEMBL7290504

SCHEMBL7290504

OC1(Cc2ccc(F)cc2)CCN(CCCOc2ccc(OCc3ccccc3)cc2)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.57
NPC1 O15118 3/20 0.57
RAB9A P51151 3/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
MAPT P10636 2/20 0.55
GRIN2D O15399 1/20 0.55
GRIN3B O60391 1/20 0.55
GRIN1 Q05586 1/20 0.55
GRIN2A Q12879 1/20 0.55
GRIN2B Q13224 1/20 0.55
GRIN2C Q14957 1/20 0.55
GRIN3A Q8TCU5 1/20 0.55
HTR1A P08908 3/20 0.53
DRD2 P14416 3/20 0.53
HTR2A P28223 3/20 0.53
HRH1 P35367 3/20 0.53
DRD3 P35462 3/20 0.53
TMEM97 Q5BJF2 2/20 0.53
SIGMAR1 Q99720 2/20 0.53
ALDH1A1 P00352 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6208225 0.94 GRIN2D (0.62) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL7294820 0.93 KDM4E (0.64) KDM4ENPC1RAB9ASMN1; SMN2MAPT
Hydrochloric Acid SCHEMBL7287564 0.88 MAPT (0.68) MAPTGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7286173 0.87 LTA4H (0.67) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL4692610 0.86 GRIN2D (0.69) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL6207790 0.86 GRIN2D (0.57) KDM4ENPC1RAB9ASMN1; SMN2MAPT
Hydrochloric Acid SCHEMBL7290147 0.85 GRIN2D (0.67) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL7289245 0.83 GRIN2D (0.79) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL7295960 0.83 GRIN2D (0.65) KDM4ENPC1RAB9ASMN1; SMN2MAPT
SCHEMBL6207263 0.83 GRIN2D (0.78) MAPTGRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0824098-B1 4-hydroxy-piperidine derivatives HOFFMANN LA ROCHE (CH) 2001-10-31 EP disclosed
US-5889026-A 4-hydroxy-piperodine derivatives HOFFMANN-LA ROCHE INC. (US) 1999-03-30 US disclosed
EP-0824098-A1 4-hydroxy-piperidine derivatives F. HOFFMANN-LA ROCHE AG (CH) 1998-02-18 EP disclosed