SCHEMBL7290900

SCHEMBL7290900

CCCCc1ccc(C(Cl)C(N)=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.54
HPGD P15428 1/20 0.54
HSD17B10 Q99714 1/20 0.54
RARB P10826 1/20 0.46
PLK1 P53350 1/20 0.46
THRA P10827 2/20 0.45
THRB P10828 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
CA2 P00918 2/20 0.45
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
CYSLTR2 Q9NS75 1/20 0.43
CYSLTR1 Q9Y271 1/20 0.43
CA1 P00915 1/20 0.43
S1PR2 O95136 1/20 0.43
S1PR1 P21453 1/20 0.43
HTR2A P28223 1/20 0.43
POLB P06746 1/20 0.43
F13A1 P00488 1/20 0.43
TGM2 P21980 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6066130 0.85 ALDH1A1 (0.56) ALDH1A1HPGDHSD17B10RARBPLK1
SCHEMBL6803238 0.78 ALDH1A1 (0.47) ALDH1A1HPGDHSD17B10RARBPLK1
SCHEMBL22571095 0.77 ALDH1A1 (0.53) ALDH1A1HPGDHSD17B10RARBPLK1
SCHEMBL7288309 0.76 MAOA (0.48) ALDH1A1HPGDPLK1THRATHRB
SCHEMBL8089660 0.76 ALDH1A1 (0.52) ALDH1A1HPGDHSD17B10RARBPLK1
SCHEMBL7282846 0.76 EPHX1 (0.69) RARBHTR2AAKR1C2
SCHEMBL9379104 0.75 ALDH1A1 (0.51) ALDH1A1HSD17B10RARBTHRATHRB
SCHEMBL11876242 0.75 PSEN1 (0.39) ALDH1A1HPGDTHRB
SCHEMBL7282009 0.74 MMP9 (0.33) HPGDCA2CA1
SCHEMBL4055722 0.74 CA2 (0.55) ALDH1A1HPGDHSD17B10RARBPLK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4567264-A ADRENERGIC BLOCKING AGENTS SYNTEX (U.S.A.) INC. (US) 1986-01-28 US disclosed
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed
US-4499100-A CARDIOUVASCULAR DISORDERS SYNTEX (U.S.A.) INC. (US) 1985-02-12 US disclosed
EP-0126449-A1 Cardioselective aryloxy- and arylthio-hydroxypropyl piperazinyl acetanilides wich affect calcium entry SYNTEX (U.S.A.) INC. (US) 1984-11-28 EP disclosed