SCHEMBL7291933

SCHEMBL7291933

Cc1ccc2[nH]cc(C(=O)OCC3CCN(CCNS(C)(=O)=O)CC3)c2c1

nearest known ligand 0.61

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 3/20 0.61
CYP2C9 P11712 2/20 0.61
PMP22 Q01453 2/20 0.61
NPSR1 Q6W5P4 2/20 0.61
CYP1A2 P05177 1/20 0.61
ALOX15 P16050 1/20 0.61
NFKB1 P19838 1/20 0.61
LMNA P02545 2/20 0.54
MEN1 O00255 1/20 0.54
CYP3A4 P08684 1/20 0.54
KMT2A Q03164 1/20 0.54
NR4A2 P43354 1/20 0.47
GSK3B P49841 1/20 0.46
HTT P42858 1/20 0.46
CARM1 Q86X55 1/20 0.43
PRMT6 Q96LA8 1/20 0.43
RAB9A P51151 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7302280 0.90 CYP2C9 (0.66) HTR4CYP2C9PMP22NPSR1CYP1A2
SCHEMBL7303858 0.88 HTR4 (0.69) HTR4CYP2C9PMP22NPSR1CYP1A2
SCHEMBL7292069 0.82 CYP2C9 (0.78) HTR4CYP2C9PMP22NPSR1CYP1A2
SCHEMBL7310046 0.76 ACHE (0.46) HTR4CYP2C9PMP22NPSR1CYP1A2
SCHEMBL1502039 0.76 HTR4 (1.00) HTR4CYP2C9PMP22NPSR1CYP1A2
SCHEMBL29397805 0.76 HTR4 (1.00) HTR4CYP2C9PMP22NPSR1CYP1A2
SCHEMBL7260342 0.75 HTR4 (0.64) HTR4CYP2C9PMP22NPSR1CYP1A2
SCHEMBL7300888 0.75 HTR4 (0.77) HTR4CYP2C9PMP22NPSR1CYP1A2
Hydrochloric Acid SCHEMBL7291228 0.74 HTR4 (0.76) HTR4CYP2C9PMP22NPSR1CYP1A2
SCHEMBL29626583 0.73 HTR4 (1.00) HTR4CYP2C9PMP22NPSR1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0501322-B1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LTD (GB) 1996-09-04 EP claimed
EP-0501322-A1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LIMITED (GB) 1992-09-02 EP claimed
EP-0501322-B1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LTD (GB) 1996-09-04 EP disclosed
WO-1992014727-A1 3-PIPERIDINYLMETHYLCARBOXYLATE SUBSTITUTED INDOLES GLAXO GROUP LIMITED (GB) 1992-09-03 WO disclosed
EP-0501322-A1 3-Piperidinylmethylcarboxylate substituted indoles GLAXO GROUP LIMITED (GB) 1992-09-02 EP disclosed