SCHEMBL7293165

SCHEMBL7293165

Nc1ccc2c(c1)CC(CC(=O)C1CCN[C@H]1C(=O)N1CCCC1)C2

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PREP P48147 14/20 0.40
BRD4 O60885 1/20 0.36
ATAD2 Q6PL18 1/20 0.36
ADAM10 O14672 3/20 0.33
ERBB2 P04626 3/20 0.33
MMP2 P08253 2/20 0.33
MC4R P32245 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7302998 0.88 DPP4 (0.42) PREPADAM10ERBB2MMP2MC4R
SCHEMBL7296377 0.88 DPP4 (0.42) PREPMC4R
SCHEMBL7292264 0.85 PNMT (0.43) PREP
SCHEMBL8154403 0.81 PREP (0.57) PREP
SCHEMBL8153717 0.81 PREP (0.57) PREP
SCHEMBL7294247 0.81 PREP (0.57) PREP
SCHEMBL7293159 0.80 PREP (0.37) PREPBRD4ATAD2
SCHEMBL7440061 0.79 CYP26A1 (0.44) PREP
SCHEMBL7303377 0.77 PREP (0.42) PREPBRD4ATAD2ADAM10ERBB2
SCHEMBL9791388 0.76 PREP (0.49) PREPADAM10ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6017929-A Cholinesterase activator ZERIA PHARMACEUTICAL CO., LTD. (JP) 2000-01-25 US disclosed
EP-0754454-A1 CHOLINESTERASE ACTIVATOR ZERIA PHARMACEUTICAL CO., LTD. (JP) 1997-01-22 EP disclosed
EP-0372484-B1 Condensed benzene derivative ZERIA PHARM CO LTD (JP) 1994-10-26 EP disclosed
US-5028604-A Cognition Activators ZERIA PHARMACEUTICAL CO., LTD. (JP) 1991-07-02 US disclosed
EP-0372484-A2 Condensed benzene derivative ZERIA PHARMACEUTICAL CO., LTD. (JP) 1990-06-13 EP disclosed