SCHEMBL7295294

SCHEMBL7295294

CC(C)n1c(N2CCC(c3c[nH]cn3)CC2)nc2ccccc21

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
ALDH1A1 P00352 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
TAAR1 Q96RJ0 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HTT P42858 1/20 0.39
HSD11B1 P28845 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9261675 0.81 CASR (0.36)
SCHEMBL9270247 0.81 ALDH1A1 (0.34) CYP1A2CYP2C9CYP2C19ALDH1A1SMN1; SMN2
SCHEMBL7294577 0.79 SLC9A1 (0.47) CYP1A2CYP2C9CYP2C19ALDH1A1SMN1; SMN2
SCHEMBL9412037 0.79 HTR2A (0.36) ALDH1A1
SCHEMBL6771824 0.74 CYP1A2 (0.56) CYP1A2CYP2C9CYP2C19ALDH1A1SMN1; SMN2
Fumaric Acid SCHEMBL9269187 0.74 ALDH1A1 (0.38) CYP1A2CYP2C9CYP2C19ALDH1A1SMN1; SMN2
Maleic Acid SCHEMBL9269178 0.74 ALDH1A1 (0.38) CYP1A2CYP2C9CYP2C19ALDH1A1SMN1; SMN2
SCHEMBL12139036 0.71 HRH3 (0.40)
SCHEMBL6428840 0.71 TRPC3 (0.60)
SCHEMBL7426131 0.70 NPC1 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507650-B1 Piperidine derivatives, their preparation and their therapeutic application SYNTHELABO (FR) 1996-05-22 EP claimed
EP-0507650-A1 Piperidine derivatives, their preparation and their therapeutic application SYNTHELABO (FR) 1992-10-07 EP claimed
EP-0507650-B1 Piperidine derivatives, their preparation and their therapeutic application SYNTHELABO (FR) 1996-05-22 EP disclosed
US-5280030-A Containing 1-benz(oxazole, thiazole or imidazole)-4-imidazole piperidine compound SYNTHELABO (FR) 1994-01-18 US disclosed
EP-0507650-A1 Piperidine derivatives, their preparation and their therapeutic application SYNTHELABO (FR) 1992-10-07 EP disclosed