SCHEMBL7297429

SCHEMBL7297429

CCn1ccnc1SCC(C)(C)[O]

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
ALDH1A1 P00352 3/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2D6 P10635 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
ALOX12 P18054 1/20 0.35
TP53 P04637 2/20 0.35
LMNA P02545 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
THRB P10828 1/20 0.34
POLB P06746 3/20 0.34
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
ALOX15B O15296 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7350391 0.83 KMT2A (0.39) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL7297435 0.73 KMT2A (0.33) KMT2AMEN1ALDH1A1SMN1; SMN2CHRM5
SCHEMBL28198306 0.69 SMN1; SMN2 (0.37) KMT2AMEN1ALDH1A1LMNASMN1; SMN2
SCHEMBL8541839 0.68 KMT2A (0.50) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL3868248 0.67 GAA (0.35) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL8465837 0.66 LMNA (0.32) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL7286212 0.66 SMN1; SMN2 (0.32) KMT2AALDH1A1SMN1; SMN2POLB
SCHEMBL19386625 0.66 EHMT2 (0.41) KMT2AMEN1ALDH1A1CYP1A2CYP3A4
SCHEMBL4687384 0.65 ALDH1A1 (0.50) KMT2AMEN1ALDH1A1TP53LMNA
SCHEMBL464563 0.65 KCNH2 (0.43) KMT2AALDH1A1CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5652247-A VASOPRESSIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD (JP) 1997-07-29 US disclosed
US-5436254-A Vaopressin antagonists OTSUKA PHARMACEUTICAL COMPANY, LTD. (JP) 1995-07-25 US disclosed
EP-0602209-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-06-22 EP disclosed
EP-0382185-B1 Carbostyril derivatives OTSUKA PHARMA CO LTD (JP) 1994-06-15 EP disclosed
WO-1994001113-A1 OXYTOCIN ANTAGONIST OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1994-01-20 WO disclosed
US-5225402-A Vasopressin antagonist, vasodilation, hypotensive, diuretics and anticoagulants OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1993-07-06 US disclosed
EP-0382185-A2 Carbostyril derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1990-08-16 EP disclosed