SCHEMBL7298709

SCHEMBL7298709

O=C(O)O[C@@H]1CCCN1C(=O)CNc1ccc(NCC(=O)N2CCC[C@@H]2C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.46
ALOX12 P18054 1/20 0.46
KMT2A Q03164 1/20 0.46
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ACE P12821 8/20 0.43
ACE2 Q9BYF1 3/20 0.42
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
UTS2R Q9UKP6 1/20 0.41
MVD P53602 2/20 0.40
DPP4 P27487 1/20 0.40
CHRM2 P08172 1/20 0.40
CHRM4 P08173 1/20 0.40
CHRM1 P11229 1/20 0.40
CHRM3 P20309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6792962 0.90 THRB (0.55) THRBALOX12KMT2AALDH1A1SMN1; SMN2
SCHEMBL5544779 0.90 THRB (0.55) THRBALOX12KMT2AALDH1A1SMN1; SMN2
SCHEMBL6438383 0.84 ACE (0.53) THRBALOX12KMT2AALDH1A1SMN1; SMN2
SCHEMBL13250828 0.84 THRB (0.49) THRBALOX12KMT2AALDH1A1SMN1; SMN2
Trifluoroacetic Acid SCHEMBL6786573 0.82 THRB (0.51) THRBALOX12KMT2AACEACE2
SCHEMBL7290822 0.81 ALDH1A1 (0.46) ALDH1A1SMN1; SMN2ACEACE2MVD
SCHEMBL6436570 0.81 ACE (0.49) THRBALOX12KMT2AALDH1A1SMN1; SMN2
SCHEMBL31710128 0.81 DGAT1 (0.53) THRBALOX12KMT2AACEACE2
SCHEMBL7288562 0.79 ALDH1A1 (0.53) KMT2AALDH1A1SMN1; SMN2MVD
SCHEMBL6786583 0.78 THRB (0.45) THRBALOX12KMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0915088-B1 D-Proline derivatives HOFFMANN LA ROCHE (CH) 2002-09-18 EP claimed