SCHEMBL7299337

SCHEMBL7299337

O=C(CCNC(=O)[C@@H]1CCNC1)OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CPB1 P15086 1/20 0.47
HTR2C P28335 2/20 0.46
GAA P10253 2/20 0.45
HTT P42858 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
F10 P00742 1/20 0.43
EPHX2 P34913 1/20 0.43
ALDH1A1 P00352 3/20 0.41
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
GLA P06280 1/20 0.41
MC4R P32245 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
USP2 O75604 1/20 0.40
HPGD P15428 1/20 0.40
ITGB3 P05106 1/20 0.40
ITGA2B P08514 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7296884 0.93 F10 (0.48) CPB1HTR2CGAAHTTMEN1
SCHEMBL1938495 0.87 LMNA (0.52) CPB1HTR2CGAAHTTMEN1
SCHEMBL2261792 0.87 LMNA (0.52) CPB1HTR2CGAAHTTMEN1
SCHEMBL1938713 0.87 LMNA (0.52) CPB1HTR2CGAAHTTMEN1
SCHEMBL10563477 0.81 ALDH1A1 (0.43) HTR2CGAAMEN1KMT2AEPHX2
SCHEMBL7659939 0.81 CPB1 (0.49) CPB1GAAHTTMEN1KMT2A
SCHEMBL1938499 0.79 SMN1; SMN2 (0.55) CPB1GAAHTTMEN1KMT2A
SCHEMBL17335891 0.79 MEN1 (0.43) CPB1HTR2CGAAHTTMEN1
Hydrochloric Acid SCHEMBL17335888 0.78 MEN1 (0.42) CPB1HTR2CGAAMEN1KMT2A
SCHEMBL2450751 0.78 ALDH1A1 (0.65) HTR2CALDH1A1MC4RUSP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0445796-B1 Derivatives of acetic acid containing peptide bonds HOFFMANN LA ROCHE (CH) 1998-06-17 EP disclosed
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed
EP-0445796-A2 Derivatives of acetic acid F. HOFFMANN-LA ROCHE AG (CH) 1991-09-11 EP disclosed