SCHEMBL7299651

SCHEMBL7299651

CCOC(=O)CCN1CCn2nc(OC(=O)OCc3ccccc3)cc2C1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.41
GRM3 Q14832 1/20 0.41
TMEM97 Q5BJF2 6/20 0.41
SIGMAR1 Q99720 6/20 0.41
SLC6A2 P23975 2/20 0.41
HRH2 P25021 2/20 0.41
HRH1 P35367 2/20 0.41
CHRM1 P11229 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
HTR1A P08908 1/20 0.39
CHRM5 P08912 1/20 0.39
ADRA1D P25100 1/20 0.39
HTR1B P28222 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
HTR1E P28566 1/20 0.39
HTR2B P41595 1/20 0.39
SLC6A3 Q01959 1/20 0.39
ALDH1A1 P00352 3/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7300441 0.95 GRM5 (0.40) GRM5GRM3TMEM97SIGMAR1SLC6A2
SCHEMBL7304398 0.85 ITGB3 (0.38) ALDH1A1PKMPOLBCYP2C19CYP1A2
SCHEMBL6475204 0.85 PKM (0.49) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL6481898 0.80 PKM (0.48) TMEM97SIGMAR1SLC6A2HRH2HRH1
SCHEMBL7314851 0.79 TNF (0.41) ALDH1A1CYP2C19CYP1A2MEN1KMT2A
SCHEMBL6474441 0.77 POLB (0.52) ALDH1A1PKMPOLBCYP2C19CYP1A2
SCHEMBL6474409 0.75 ITGB3 (0.46) PKMSMN1; SMN2
SCHEMBL6474034 0.71 POLB (0.50) ALDH1A1PKMPOLBCYP2C19CYP1A2
SCHEMBL6480916 0.71 ITGB3 (0.47) SMN1; SMN2
SCHEMBL7678810 0.71 SMN1; SMN2 (0.44) PKMSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0854140-B1 Vitronectin receptor antagonists, their production and their use SANOFI AVENTIS DEUTSCHLAND (DE) 2013-11-06 EP disclosed
EP-0854140-A2 Vitronectin receptor antagonists, their production and their use HOECHST AKTIENGESELLSCHAFT (DE) 1998-07-22 EP disclosed